SCHEMBL5686342

SCHEMBL5686342

CCC[C@H]1CC[C@@H]2c3ccc(OS(=O)(=O)C(F)(F)F)cc3CC[C@H]2[C@@H]1F

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.46
HTR1D P28221 1/20 0.46
DRD3 P35462 1/20 0.46
AKR1C3 P42330 1/20 0.43
STS P08842 10/20 0.41
ABCC4 O15439 3/20 0.40
ABCC1 P33527 2/20 0.40
KDM4E B2RXH2 2/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA9 Q16790 2/20 0.40
CYP2C9 P11712 1/20 0.40
SLCO1B1 Q9Y6L6 1/20 0.40
ESR1 P03372 1/20 0.40
CA4 P22748 1/20 0.40
CA6 P23280 1/20 0.40
ESR2 Q92731 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5686345 1.00 DRD2 (0.46) DRD2HTR1DDRD3AKR1C3STS
SCHEMBL5683918 0.79 STS (0.50) STSCYP2C9ESR1ESR2
SCHEMBL5683915 0.79 STS (0.50) STSCYP2C9ESR1ESR2
SCHEMBL5686598 0.78 DRD2 (0.47) DRD2HTR1DDRD3AKR1C3
SCHEMBL5686604 0.78 DRD2 (0.47) DRD2HTR1DDRD3AKR1C3
SCHEMBL7530599 0.74 STS (0.43) DRD2STS
SCHEMBL27051298 0.71 STS (0.54) AKR1C3STSABCC4ABCC1
SCHEMBL12054334 0.71 STS (0.77) STSABCC4ABCC1KDM4ECA1
SCHEMBL31321077 0.71 STS (0.77) STSABCC4ABCC1KDM4ECA1
SCHEMBL3825597 0.71 STS (0.77) STSABCC4ABCC1KDM4ECA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7067179-B1 Fused ring compound DAINIPPON INK AND CHEMICALS, INC. (JP) 2006-06-27 US disclosed
EP-1201632-B1 FUSED RING COMPOUND DAINIPPON INK & CHEMICALS (JP) 2006-03-29 EP disclosed
EP-1201632-A1 FUSED RING COMPOUND DAINIPPON INK AND CHEMICALS, INC. (JP) 2002-05-02 EP disclosed