SCHEMBL5688359

SCHEMBL5688359

CC(=O)Nc1cccc(-c2ccc(C(O)(c3c[nH]cn3)C(C)C)cc2)c1C

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 11/20 0.43
CYP3A4 P08684 6/20 0.43
KDM4E B2RXH2 1/20 0.37
BTK Q06187 2/20 0.36
TOP2A P11388 1/20 0.35
PARP14 Q460N5 1/20 0.35
CCNE2 O96020 2/20 0.34
CCNE1 P24864 2/20 0.34
CDK2 P24941 2/20 0.34
CDK4 P11802 1/20 0.34
CCND1 P24385 1/20 0.34
FFAR2 O15552 1/20 0.34
MAOA P21397 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22284881 0.82 CYP17A1 (0.34) CYP17A1CYP3A4
SCHEMBL5688374 0.81 CYP17A1 (0.63) CYP17A1CYP3A4
SCHEMBL7563594 0.81 CYP17A1 (0.66) CYP17A1CYP3A4
SCHEMBL5688564 0.81 CYP17A1 (0.66) CYP17A1CYP3A4
SCHEMBL22284897 0.80 LRRK2 (0.41) CYP17A1CYP3A4
SCHEMBL5689388 0.79 CYP17A1 (0.39) CYP17A1CYP3A4TOP2A
SCHEMBL5688618 0.79 CYP17A1 (0.46) CYP17A1CYP3A4BTK
SCHEMBL5688682 0.79 CYP17A1 (0.67) CYP17A1CYP3A4
SCHEMBL5690780 0.78 CYP17A1 (0.49) CYP17A1CYP3A4MAOA
SCHEMBL5688810 0.78 FFAR2 (0.37) CYP17A1CYP3A4KDM4EFFAR2MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1227086-B1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2006-03-29 EP disclosed
US-6518257-B1 1-substituted phenyl-1-(1h-imidazol-4-yl) alcohols, process for producing the same and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-02-11 US disclosed
EP-1227086-A1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-07-31 EP disclosed