SCHEMBL5688382

SCHEMBL5688382

CNC(=O)c1cccc(-c2ccc(C(C)(O)c3cn(C(c4ccccc4)(c4ccccc4)c4ccccc4)cn3)cc2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 2/20 0.45
CYP3A4 P08684 2/20 0.45
NR4A2 P43354 2/20 0.39
PIK3CG P48736 1/20 0.39
CDK8 P49336 1/20 0.39
PDK2 Q15119 1/20 0.39
ATM Q13315 1/20 0.39
KDM5A P29375 1/20 0.39
KDM4C Q9H3R0 1/20 0.39
KDM5B Q9UGL1 1/20 0.39
KIF11 P52732 1/20 0.39
CRBN Q96SW2 1/20 0.39
HDAC8 Q9BY41 1/20 0.38
ACSS2 Q9NR19 1/20 0.37
POLB P06746 1/20 0.37
MAPT P10636 1/20 0.37
CTDSP1 Q9GZU7 1/20 0.37
GRM5 P41594 1/20 0.36
ADRA2A P08913 1/20 0.36
ADRA1A P35348 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5689045 0.88 CYP17A1 (0.43) CYP17A1CYP3A4NR4A2PIK3CGCDK8
SCHEMBL5688583 0.88 CYP17A1 (0.56) CYP17A1CYP3A4NR4A2PIK3CGCDK8
SCHEMBL5688876 0.85 CYP17A1 (0.41) CYP17A1CYP3A4NR4A2PIK3CGCDK8
SCHEMBL4025339 0.84 CYP17A1 (0.53) CYP17A1CYP3A4KIF11ACSS2
SCHEMBL5688570 0.83 CYP17A1 (0.48) CYP17A1CYP3A4NR4A2PIK3CGCDK8
SCHEMBL5689071 0.82 CYP17A1 (0.52) CYP17A1CYP3A4FYN
SCHEMBL5691363 0.79 CYP3A4 (0.46) CYP17A1CYP3A4ACSS2
SCHEMBL5691427 0.78 CYP17A1 (0.42) CYP17A1CYP3A4RXRARXRB
SCHEMBL5688802 0.78 CYP17A1 (0.45) CYP17A1CYP3A4CDK8ACSS2
SCHEMBL5688388 0.77 SIRT2 (0.46) CYP17A1CYP3A4PIK3CGCDK8KDM5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1227086-B1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2006-03-29 EP disclosed
US-6518257-B1 1-substituted phenyl-1-(1h-imidazol-4-yl) alcohols, process for producing the same and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-02-11 US disclosed
EP-1227086-A1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-07-31 EP disclosed