SCHEMBL5688570

SCHEMBL5688570

CNC(=O)c1cccc(-c2cccc(C(O)(c3cn(C(c4ccccc4)(c4ccccc4)c4ccccc4)cn3)C(C)C)c2)c1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 5/20 0.48
CYP3A4 P08684 5/20 0.48
CDK8 P49336 1/20 0.39
KDM5A P29375 1/20 0.38
KDM4C Q9H3R0 1/20 0.38
KDM5B Q9UGL1 1/20 0.38
KIF11 P52732 1/20 0.38
FYN P06241 1/20 0.37
ACSS2 Q9NR19 2/20 0.37
PIK3CG P48736 1/20 0.37
NR4A2 P43354 1/20 0.37
SIRT2 Q8IXJ6 4/20 0.36
PDK2 Q15119 1/20 0.36
ADRA2A P08913 1/20 0.36
ADRA1A P35348 1/20 0.36
FGFR1 P11362 1/20 0.36
FGFR3 P22607 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5688583 0.94 CYP17A1 (0.56) CYP17A1CYP3A4CDK8KDM5AKDM4C
SCHEMBL4031099 0.86 CYP17A1 (0.52) CYP17A1CYP3A4ACSS2SIRT2
SCHEMBL5691363 0.86 CYP3A4 (0.46) CYP17A1CYP3A4ACSS2SIRT2
SCHEMBL5688704 0.85 CYP17A1 (0.44) CYP17A1CYP3A4CDK8KDM5AKDM4C
SCHEMBL5688802 0.84 CYP17A1 (0.45) CYP17A1CYP3A4CDK8ACSS2SIRT2
SCHEMBL5688616 0.84 CYP17A1 (0.43) CYP17A1CYP3A4CDK8FYNSIRT2
SCHEMBL5690727 0.83 CYP17A1 (0.47) CYP17A1CYP3A4FYN
SCHEMBL5688382 0.83 CYP17A1 (0.45) CYP17A1CYP3A4CDK8KDM5AKDM4C
SCHEMBL5688555 0.83 CYP17A1 (0.48) CYP17A1CYP3A4PIK3CGFGFR1FGFR3
SCHEMBL5688655 0.83 CYP17A1 (0.44) CYP17A1CYP3A4ACSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1227086-B1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2006-03-29 EP disclosed
US-6518257-B1 1-substituted phenyl-1-(1h-imidazol-4-yl) alcohols, process for producing the same and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-02-11 US disclosed
EP-1227086-A1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-07-31 EP disclosed