SCHEMBL5688583

SCHEMBL5688583

CNC(=O)c1cccc(-c2ccc(C(O)(c3cn(C(c4ccccc4)(c4ccccc4)c4ccccc4)cn3)C(C)C)cc2)c1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 10/20 0.56
CYP3A4 P08684 9/20 0.56
PIK3CG P48736 1/20 0.38
NR4A2 P43354 1/20 0.38
CDK8 P49336 1/20 0.37
PDK2 Q15119 1/20 0.37
ATM Q13315 1/20 0.37
SIRT2 Q8IXJ6 1/20 0.37
KDM5A P29375 1/20 0.37
KDM4C Q9H3R0 1/20 0.37
KDM5B Q9UGL1 1/20 0.37
ADRA2A P08913 1/20 0.37
ADRA1A P35348 1/20 0.37
KIF11 P52732 1/20 0.37
CRBN Q96SW2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5688570 0.94 CYP17A1 (0.48) CYP17A1CYP3A4PIK3CGNR4A2CDK8
SCHEMBL5691363 0.92 CYP3A4 (0.46) CYP17A1CYP3A4SIRT2
SCHEMBL5688616 0.91 CYP17A1 (0.43) CYP17A1CYP3A4CDK8SIRT2
SCHEMBL5688802 0.90 CYP17A1 (0.45) CYP17A1CYP3A4CDK8SIRT2
SCHEMBL5688555 0.89 CYP17A1 (0.48) CYP17A1CYP3A4PIK3CG
SCHEMBL5688704 0.89 CYP17A1 (0.44) CYP17A1CYP3A4CDK8ATMSIRT2
SCHEMBL5688655 0.89 CYP17A1 (0.44) CYP17A1CYP3A4
SCHEMBL5688382 0.88 CYP17A1 (0.45) CYP17A1CYP3A4PIK3CGNR4A2CDK8
SCHEMBL5690923 0.86 CYP17A1 (0.41) CYP17A1CYP3A4ATMSIRT2
SCHEMBL5689045 0.85 CYP17A1 (0.43) CYP17A1CYP3A4PIK3CGNR4A2CDK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1227086-B1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2006-03-29 EP disclosed
US-6518257-B1 1-substituted phenyl-1-(1h-imidazol-4-yl) alcohols, process for producing the same and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-02-11 US disclosed
EP-1227086-A1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-07-31 EP disclosed