SCHEMBL5688981

SCHEMBL5688981

CNC(=O)c1cccc(-c2ccc(C(O)(c3c[nH]cn3)C(C)C)cc2)n1

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 9/20 0.45
CYP3A4 P08684 6/20 0.44
CNR2 P34972 7/20 0.41
CNR1 P21554 3/20 0.41
PIM1 P11309 1/20 0.40
PIM2 Q9P1W9 1/20 0.40
SCN9A Q15858 2/20 0.39
CTSA P10619 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5688705 0.91 CYP17A1 (0.44) CYP17A1CYP3A4CNR2CNR1SCN9A
SCHEMBL5689203 0.89 CYP17A1 (0.45) CYP17A1CYP3A4CNR2SCN9ACTSA
SCHEMBL5688682 0.82 CYP17A1 (0.67) CYP17A1CYP3A4CNR2CNR1SCN9A
SCHEMBL5688304 0.80 CYP17A1 (0.68) CYP17A1CYP3A4
SCHEMBL5688557 0.80 CYP17A1 (0.51) CYP17A1CYP3A4
SCHEMBL5688460 0.78 KDM4E (0.47) CYP17A1CYP3A4
SCHEMBL5688786 0.77 CNR2 (0.44) CYP17A1CYP3A4CNR2CNR1SCN9A
SCHEMBL18770487 0.77 CYP17A1 (0.63) CYP17A1CYP3A4
SCHEMBL4024772 0.76 CYP17A1 (0.51) CYP17A1CYP3A4
SCHEMBL5688807 0.76 CYP17A1 (0.56) CYP17A1CYP3A4PIM1PIM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1227086-B1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2006-03-29 EP disclosed
US-6518257-B1 1-substituted phenyl-1-(1h-imidazol-4-yl) alcohols, process for producing the same and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-02-11 US disclosed
EP-1227086-A1 1-SUBSTITUTED PHENYL-1-(1H-IMIDAZOL-4-YL) ALCOHOLS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-07-31 EP disclosed