SCHEMBL5690282

SCHEMBL5690282

CCN(c1ccc(CC=C=O)cc1)c1nc(N)c2ncn([C@@H]3O[C@H](C(O)N(C=O)CC)[C@@H](O)[C@H]3O)c2n1

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 8/20 0.39
ADORA2A P29274 8/20 0.39
ADORA1 P30542 8/20 0.39
ADORA2B P29275 6/20 0.39
HSP90B1 P14625 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5689446 0.87 ADORA3 (0.40) ADORA3ADORA2AADORA1ADORA2B
SCHEMBL940189 0.85 ADORA2A (0.55) ADORA3ADORA2AADORA1ADORA2B
SCHEMBL258935 0.78 ADORA3 (0.59) ADORA3ADORA2AADORA1ADORA2B
SCHEMBL177772 0.75 AHCY (0.61) ADORA3ADORA2AADORA1ADORA2BHSP90B1
SCHEMBL28901883 0.75 AHCY (0.61) ADORA3ADORA2AADORA1ADORA2BHSP90B1
SCHEMBL29877256 0.75 AHCY (0.61) ADORA3ADORA2AADORA1ADORA2BHSP90B1
SCHEMBL2295172 0.75 ADORA2A (0.65) ADORA3ADORA2AADORA1ADORA2B
SCHEMBL8102781 0.75 ADORA2A (0.64) ADORA3ADORA2AADORA1ADORA2B
SCHEMBL1081737 0.74 ADORA2A (0.68) ADORA3ADORA2AADORA1ADORA2B
SCHEMBL5964576 0.74 ADORA3 (0.67) ADORA3ADORA2AADORA1ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060205671-A1 Compositions and methods for use of a protease inhibitor and adenosine for preventing organ ischemia and reperfusion injury EMORY UNIVERSITY 2006-09-14 US claimed
EP-1638579-A2 COMPOSITIONS AND METHODS FOR USE OF A PROTEASE INHIBITOR AND ADENOSINE FOR PREVENTING ORGAN ISCHEMIA AND REPERFUSION INJURY EMORY UNIVERSITY (US) 2006-03-29 EP claimed
WO-2005003150-A2 COMPOSITIONS AND METHODS FOR USE OF A PROTEASE INHIBITOR AND ADENOSINE FOR PREVENTING ORGAN ISCHEMIA AND REPERFUSION INJURY EMORY UNIVERSITY (US) 2005-01-13 WO claimed
US-20060205671-A1 Compositions and methods for use of a protease inhibitor and adenosine for preventing organ ischemia and reperfusion injury EMORY UNIVERSITY 2006-09-14 US disclosed
EP-1638579-A2 COMPOSITIONS AND METHODS FOR USE OF A PROTEASE INHIBITOR AND ADENOSINE FOR PREVENTING ORGAN ISCHEMIA AND REPERFUSION INJURY EMORY UNIVERSITY (US) 2006-03-29 EP disclosed
WO-2005003150-A2 COMPOSITIONS AND METHODS FOR USE OF A PROTEASE INHIBITOR AND ADENOSINE FOR PREVENTING ORGAN ISCHEMIA AND REPERFUSION INJURY EMORY UNIVERSITY (US) 2005-01-13 WO disclosed