SCHEMBL5691985

SCHEMBL5691985

CC(CC(=O)O)c1ccc(N)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 6/20 0.59
POLB P06746 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
ACHE P22303 1/20 0.46
ALDH1A1 P00352 2/20 0.44
GRIA4 P48058 1/20 0.42
TSHR P16473 2/20 0.42
STAT3 P40763 1/20 0.42
USP5 P45974 1/20 0.42
FFAR4 Q5NUL3 1/20 0.41
GABBR2 O75899 4/20 0.41
GABBR1 Q9UBS5 4/20 0.41
LMNA P02545 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP3A4 P08684 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
NFKB1 P19838 1/20 0.41
DRD3 P35462 1/20 0.41
BLM P54132 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5691981 1.00 FFAR1 (0.59) FFAR1POLBSMN1; SMN2TDP1ACHE
SCHEMBL11332403 0.88 FFAR1 (0.62) FFAR1POLBSMN1; SMN2ACHEALDH1A1
SCHEMBL12883299 0.84 ACHE (0.46) FFAR1POLBSMN1; SMN2TDP1ACHE
SCHEMBL27953749 0.82 FFAR1 (0.41) FFAR1POLBSMN1; SMN2TDP1ACHE
SCHEMBL25152959 0.82 ACHE (0.67) FFAR1POLBACHEALDH1A1TSHR
SCHEMBL7559049 0.82 ACHE (0.67) FFAR1POLBACHEALDH1A1TSHR
SCHEMBL12883165 0.82 ACHE (0.67) FFAR1POLBACHEALDH1A1TSHR
SCHEMBL31522488 0.82 FFAR1 (0.61) FFAR1TDP1ACHEALDH1A1TSHR
SCHEMBL1162528 0.82 FFAR1 (0.61) FFAR1TDP1ACHEALDH1A1TSHR
SCHEMBL13140496 0.82 FFAR1 (0.61) FFAR1TDP1ACHEALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019168654-A9 DNA-TEMPLATED MACROCYCLE LIBRARY PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2019-10-17 WO disclosed
CN-108530333-A A kind of preparation method of 4- phenyl -2-Pyrrolidone 杭州卢普生物科技有限公司 2018-09-14 CN disclosed
EP-2310371-B1 PPAR AGONIST COMPOUNDS AND PREPARATION AND USES THEREOF FOR TREATING DIABETES AND/OR DYSLIPIDEMIA GENFIT (FR) 2013-05-15 EP disclosed
CN-101633625-B Method for preparing R-beta-aminobenzene butyric acid derivative JIANGSU HENGRUI MEDICINE CO 2013-02-13 CN disclosed
CN-102115450-A Preparation method for 4-amino-3-phenylbutyric acid SHANGHAI SEPAL CHEMICAL CO LTD 2011-07-06 CN disclosed
EP-1153017-B1 BICYCLIC COMPOUNDS AND THEIR USE AS INTEGRIN RECEPTOR LIGANDS AVENTIS PHARMA LTD (GB) 2006-05-03 EP disclosed
US-6593354-B2 Amide substituted benzimidazole or benzoxazole; regulating the interaction of vascular cell adhesion molecule-1 and fibronectin with the integrin vascular cell adhesion molecule very late antigen-4 AVENTIS PHARMA LIMITED (GB) 2003-07-15 US disclosed
US-20020137782-A1 Substituted bicyclic compounds AVENTIS PHARMA LIMITED (GB) 2002-09-26 US disclosed
EP-1153017-A1 BICYCLIC COMPOUNDS AND THEIR USE AS INTEGRIN RECEPTOR LIGANDS Aventis Pharma Limited (GB) 2001-11-14 EP disclosed
WO-2000049005-A1 BICYCLIC COMPOUNDS AND THEIR USE AS INTEGRIN RECEPTOR LIGANDS AVENTIS PHARMA LIMITED (GB) 2000-08-24 WO disclosed
EP-0554023-B1 Corrosion inhibitors CIBA GEIGY AG (CH) 1997-04-23 EP disclosed
US-5250325-A Corrosion inhibitors CIBA-GEIGY CORPORATION (US) 1993-10-05 US disclosed
EP-0554023-A1 Corrosion inhibitors CIBA-GEIGY AG (CH) 1993-08-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020137782-A1 Substituted bicyclic compounds ITGA1, VCAM1, ITGB1 FFAR1 175/4885POLB 3796/4885SMN1; SMN2 2427/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.