SCHEMBL7049149

SCHEMBL7049149

NCc1nc(NCCc2ccccc2)c2ncn([C@@H]3O[C@H](CO)[C@@H](O)[C@H]3O)c2n1

nearest known ligand 0.79

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PGK1 P00558 4/20 0.79
PGK2 P07205 4/20 0.79
ADORA3 P0DMS8 6/20 0.73
ADORA1 P30542 5/20 0.73
ADORA2A P29274 4/20 0.73
TSHR P16473 2/20 0.73
NFKB1 P19838 1/20 0.73
THPO P40225 1/20 0.73
LMNA P02545 1/20 0.63
MAPT P10636 1/20 0.63
NPSR1 Q6W5P4 1/20 0.63
CYP3A4 P08684 1/20 0.63
MAPK1 P28482 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1120648 0.91 ADORA3 (0.72) PGK1PGK2ADORA3ADORA1ADORA2A
SCHEMBL7771098 0.90 PGK1 (0.64) PGK1PGK2ADORA3ADORA1ADORA2A
SCHEMBL5694952 0.90 PGK1 (0.64) PGK1PGK2ADORA3ADORA1ADORA2A
SCHEMBL31201331 0.87 ADORA1 (0.88) PGK1PGK2ADORA3ADORA1ADORA2A
SCHEMBL5414368 0.86 ADORA2A (0.72) ADORA3ADORA1ADORA2A
SCHEMBL6328801 0.86 PGK1 (0.71) PGK1PGK2ADORA3ADORA1ADORA2A
SCHEMBL6328795 0.86 PGK1 (0.71) PGK1PGK2ADORA3ADORA1ADORA2A
SCHEMBL1120606 0.85 CYP1A2 (0.71) ADORA3ADORA1ADORA2ATSHRNFKB1
SCHEMBL1054862 0.84 ADORA3 (1.00) PGK1PGK2ADORA3ADORA1ADORA2A
SCHEMBL1054866 0.84 ADORA3 (1.00) PGK1PGK2ADORA3ADORA1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1220863-B1 PURINE DERIVATIVES PFIZER LTD (GB) 2003-04-23 EP disclosed
US-6350735-B1 Purine derivatives PFIZER INC 2002-02-26 US disclosed