SCHEMBL5698706

SCHEMBL5698706

FC(F)(F)c1cc(-c2cc(Cl)ccc2Cl)n(-c2ccc(S)cc2)n1

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 13/20 0.59
PTGS1 P23219 12/20 0.59
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C9 P11712 1/20 0.50
TSHR P16473 1/20 0.50
CYP2C19 P33261 1/20 0.50
THPO P40225 1/20 0.50
BLM P54132 1/20 0.50
PMP22 Q01453 1/20 0.50
HIF1A Q16665 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
PDPK1 O15530 4/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5674345 0.83 PTGS2 (0.83) PTGS2PTGS1CYP2C9PDPK1
SCHEMBL5694394 0.83 PTGS2 (0.86) PTGS2PTGS1CYP1A2CYP3A4CYP2C9
SCHEMBL5674641 0.82 PTGS2 (0.58) PTGS2PTGS1CYP1A2CYP3A4CYP2C9
Carbamic Acid SCHEMBL5858404 0.81 PTGS2 (0.57) PTGS2PTGS1PDPK1
SCHEMBL7113078 0.75 PTGS2 (1.00) PTGS2PTGS1CYP1A2CYP3A4CYP2C9
SCHEMBL6266521 0.74 PTGS1 (0.80) PTGS2PTGS1CYP2C9PDPK1
SCHEMBL3246957 0.73 PTGS2 (1.00) PTGS2PTGS1CYP2C9PDPK1
SCHEMBL8917353 0.73 PTGS2 (0.68) PTGS2PTGS1CYP1A2CYP3A4CYP2C9
SCHEMBL19205691 0.73 PTGS2 (0.74) PTGS2PTGS1PDPK1
SCHEMBL5859292 0.72 PTGS2 (0.71) PTGS2PTGS1CYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1682143-A2 COMBINATIONS COMPRISING AN HSP90 INHIBITOR AND A PHOPHODIESTERASE INHIBITOR FOR TREATING OR PREVENTING NEOPLASIA Pharmacia Corporation (US) 2006-07-26 EP disclosed
WO-2005041879-A2 COMBINATIONS COMPRISING AN Hsp90 INHIBITOR AND A PHOPHODIESTERASE INHIBITOR FOR TREATING OR PREVENTING NEOPLASIA PHARMACIA CORPORATION (US) 2005-05-12 WO disclosed