SCHEMBL5700487

SCHEMBL5700487

Cc1cccnc1S(C)(=O)=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.45
NOS1 P29475 1/20 0.45
NOS2 P35228 1/20 0.45
KMT2A Q03164 2/20 0.43
PLAU P00749 1/20 0.41
PAX8 Q06710 2/20 0.40
PTGS2 P35354 2/20 0.38
PTGS1 P23219 1/20 0.38
SLC40A1 Q9NP59 1/20 0.37
KDM4E B2RXH2 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
CYP2A6 P11509 1/20 0.37
ALOX15 P16050 1/20 0.37
HTT P42858 1/20 0.37
GLO1 Q04760 1/20 0.37
HSD11B1 P28845 1/20 0.36
FDPS P14324 1/20 0.36
NFE2L2 Q16236 1/20 0.36
TDP2 O95551 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20157296 0.83 NOS3 (0.42) NOS3NOS1NOS2KMT2APLAU
SCHEMBL20149755 0.83 NOS3 (0.42) NOS3NOS1NOS2KMT2APLAU
SCHEMBL1039344 0.81 NOS3 (0.43) NOS3NOS1NOS2KMT2APLAU
SCHEMBL3636398 0.81 NOS3 (0.48) NOS3NOS1NOS2KMT2APLAU
SCHEMBL4998230 0.81 KDM4E (0.45) NOS3NOS1NOS2KMT2APLAU
Hydrochloric Acid SCHEMBL27558535 0.79 KDM4E (0.44) NOS3NOS1NOS2KMT2APLAU
SCHEMBL31527719 0.79 KMT2A (0.49) NOS3NOS1NOS2KMT2APLAU
SCHEMBL10833748 0.78 MAPK1 (0.41) KMT2APAX8PTGS2PTGS1KDM4E
SCHEMBL2645585 0.78 KMT2A (0.40) KMT2APAX8PTGS2PTGS1KDM4E
SCHEMBL24351473 0.78 NOS3 (0.41) NOS3NOS1NOS2KMT2APLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023191953-A1 PNICTOGEN-CONTAINING HETEROCYCLIC COMPOUNDS AND THEIR USE UNIVERSITY OF RHODE ISLAND BOARD OF TRUSTEES (US) 2023-10-05 WO disclosed
US-9394302-B2 Inhibitors of influenza viruses replication VERTEX PHARMACEUTICALS INCORPORATED (US) 2016-07-19 US disclosed
US-20150191468-A1 INHIBITORS OF INFLUENZA VIRUSES REPLICATION VERTEX PHARMACEUTICALS INCORPORATED 2015-07-09 US disclosed
US-8993598-B2 Pyrrole compounds TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2015-03-31 US disclosed
US-8969387-B2 Pyrrole compounds TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2015-03-03 US disclosed
EP-2794600-A1 DIHYDRO-BENZO-OXAZINE AND DIHYDRO-PYRIDO-OXAZINE DERIVATIVES Novartis AG (CH) 2014-10-29 EP disclosed
US-20140031393-A1 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2014-01-30 US disclosed
CN-101248048-B Imidazole based LXR modulators EXELIXIS INC 2013-08-28 CN disclosed
CN-101248049-B Imidazole based lxr modulators EXELIXIS INC 2013-08-28 CN disclosed
WO-2013093849-A1 DIHYDRO-BENZO-OXAZINE AND DIHYDRO-PYRIDO-OXAZINE DERIVATIVES NOVARTIS AG (CH) 2013-06-27 WO disclosed
US-20110172275-A1 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-07-14 US disclosed
US-20110172275-A1 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-07-14 US disclosed
US-20100056577-A1 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-03-04 US disclosed
CN-101248049-A Imidazole based LXR modulators EXELIXIS INC (US) 2008-08-20 CN disclosed
CN-101248048-A Imidazole based LXR modulators EXELIXIS INC (US) 2008-08-20 CN disclosed
EP-1270582-B1 TRIPHENYLPHOSPHINE DERIVATIVES, PALLADIUM OR NICKEL COMPLEXES THEREOF, AND PROCESS FOR PREPARING BIARYL DERIVATIVES MITSUBISHI RAYON CO (JP) 2006-08-30 EP disclosed
US-6693210-B2 USING PALLADIUM, NICKEL PHOSPHINE COMPLEX AS CATALYSTS MITSUBISHI RAYON CO., LTD. (JP) 2004-02-17 US disclosed
US-20030065208-A1 Using palladium, nickel phosphine complex as catalysts MITSUBISHI RAYON CO., LTD. (JP) 2003-04-03 US disclosed
EP-1270582-A1 TRIPHENYLPHOSPHINE DERIVATIVE, PRODUCTION PROCESS THEREFOR, PALLADIUM COMPLEX THEREOF, AND PROCESS FOR PRODUCING BIARYL DERIVATIVE Mitsubishi Rayon Co., Ltd. (JP) 2003-01-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100056577-A1 PYRROLE COMPOUNDS PRLHR, C1R, C1S NOS3 1334/4885NOS1 2085/4885NOS2 1956/4885
US-20140031393-A1 PYRROLE COMPOUNDS PRLHR, C1R, C1S NOS3 1334/4885NOS1 2085/4885NOS2 1956/4885
US-20030065208-A1 Using palladium, nickel phosphine complex as catalysts PDCD1LG2, PIK3CA, PDCD1 NOS3 3395/4885NOS1 3878/4885NOS2 3241/4885
US-20110172275-A1 PYRROLE COMPOUNDS PRLHR, C1R, C1S NOS3 1334/4885NOS1 2085/4885NOS2 1956/4885
US-20150191468-A1 INHIBITORS OF INFLUENZA VIRUSES REPLICATION ACE, RNASEH1, ACE2 NOS3 3318/4885NOS1 2467/4885NOS2 2626/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.