SCHEMBL5704141

SCHEMBL5704141

COC(=O)c1ccc(-c2ccc(CCNC(Cc3ccccc3)[C@H](O)c3ccccc3)cc2)cc1[N+](=O)[O-]

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 16/20 0.49
ADRB1 P08588 12/20 0.49
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
ABCB1 P08183 1/20 0.40
ADRB2 P07550 1/20 0.39
APP P05067 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5703739 0.83 ADRB3 (0.56) ADRB3ADRB1ADRB2
SCHEMBL5703738 0.83 ADRB3 (0.49) ADRB3ADRB1ADRB2
SCHEMBL4584637 0.78 L3MBTL1 (0.42) ADRB3ADRB1ABCB1ADRB2APP
SCHEMBL4584644 0.78 L3MBTL1 (0.42) ADRB3ADRB1ABCB1ADRB2APP
SCHEMBL6269328 0.76 KDM4E (0.41) ADRB3ADRB1RAB9AADRB2
SCHEMBL2271534 0.76 ABCB1 (0.61) ABCB1
SCHEMBL6272979 0.74 POLB (0.41) NPC1RAB9A
SCHEMBL4584322 0.71 L3MBTL1 (0.49) NPC1RAB9AABCB1
SCHEMBL6590093 0.69 ERN1 (0.46) ABCB1
SCHEMBL2277745 0.69 PDGFRB (0.46) NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1697301-A2 AMINOALCOHOL DERIVATIVES Astellas Pharma Inc. (JP) 2006-09-06 EP disclosed
WO-2005061433-A2 AMINOALCOHOL DERIVATIVES ASTELLAS PHARMA INC. (JP) 2005-07-07 WO disclosed