SCHEMBL570435

SCHEMBL570435

OC1O[C@@H](C2CC2)[C@@H](O)[C@@H](O)[C@@H]1O

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 2/20 0.43
ALDH1A1 P00352 2/20 0.30
TSHR P16473 2/20 0.30
LMNA P02545 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23903725 0.77 LGALS3 (0.47) ALDH1A1TSHRLMNATDP1
SCHEMBL9613597 0.69 GBA1 (0.47) GBA1LMNA
SCHEMBL16812686 0.69 GBA1 (0.47) GBA1LMNA
SCHEMBL12017371 0.69 GBA1 (0.47) GBA1LMNA
SCHEMBL10076292 0.69 GBA1 (0.47) GBA1LMNA
SCHEMBL11915509 0.69 GBA1 (0.47) GBA1LMNA
SCHEMBL14191362 0.69 GBA1 (0.47) GBA1LMNA
SCHEMBL14191363 0.69 GBA1 (0.47) GBA1LMNA
SCHEMBL22043674 0.69 GBA1 (0.47) GBA1LMNA
SCHEMBL16550452 0.69 GBA1 (0.47) GBA1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2282773-B2 METHODS AND COMPOSITIONS FOR MAKING ANTIBODIES AND ANTIBODY DERIVATIVES WITH REDUCED CORE FUCOSYLATION SEAGEN INC (US) 2025-03-05 EP disclosed
US-20230055475-A1 METHODS AND COMPOSITIONS FOR MAKING ANTIBODIES AND ANTIBODY DERIVATIVES WITH REDUCED CORE FUCOSYLATION SEAGEN INC (US) 2023-02-23 US disclosed
US-11319526-B2 Methods and compositions for making antibodies and antibody derivatives with reduced core fucosylation SEAGEN INC. (US) 2022-05-03 US disclosed
US-11033561-B2 Methods of inhibition of protein fucosylation in vivo using fucose analogs SEAGEN INC. (US) 2021-06-15 US disclosed
US-20200061091-A1 METHODS OF INHIBITION OF PROTEIN FUCOSYLATION IN VIVO USING FUCOSE ANALOGS SEATTLE GENETICS, INC. (US) 2020-02-27 US disclosed
US-10443035-B2 Methods and compositions for making antibodies and antibody derivatives with reduced core fucosylation SEATTLE GENETICS, INC. (US) 2019-10-15 US disclosed
US-20190276796-A1 METHODS AND COMPOSITIONS FOR MAKING ANTIBODIES AND ANTIBODY DERIVATIVES WITH REDUCED CORE FUCOSYLATION SEAGEN INC. 2019-09-12 US disclosed
EP-3513794-A2 FUCOSE ANALOGS FOR INHIBITION OF PROTEIN FUCOSYLATION IN VIVO Seattle Genetics, Inc. (US) 2019-07-24 EP disclosed
US-10342811-B2 Methods of inhibition of protein fucosylation in vivo using fucose analogs SEATTLE GENETICS, INC. (US) 2019-07-09 US disclosed
EP-2608796-B1 INHIBITION OF PROTEIN FUCOSYLATION IN VIVO USING FUCOSE ANALOGS SEATTLE GENETICS INC (US) 2018-11-21 EP disclosed
US-8993326-B2 Methods and compositions for making antibodies and antibody derivatives with reduced core fucosylation SEATTLE GENETICS, INC. (US) 2015-03-31 US disclosed
US-20140031536-A1 METHODS AND COMPOSITIONS FOR MAKING ANTIBODIES AND ANTIBODY DERIVATIVES WITH REDUCED CORE FUCOSYLATION SEATTLE GENETICS, INC. (US) 2014-01-30 US disclosed
EP-2282773-B1 METHODS AND COMPOSITIONS FOR MAKING ANTIBODIES AND ANTIBODY DERIVATIVES WITH REDUCED CORE FUCOSYLATION SEATTLE GENETICS INC (US) 2014-01-15 EP disclosed
US-8574907-B2 Methods and compositions for making antibodies and antibody derivatives with reduced core fucosylation SEATTLE GENETICS, INC. (US) 2013-11-05 US disclosed
EP-2608796-A2 METHODS OF INHIBITION OF PROTEIN FUCOSYLATION IN VIVO USING FUCOSE ANALOGS Seattle Genetics, Inc. (US) 2013-07-03 EP disclosed
US-20130129784-A1 METHODS OF INHIBITION OF PROTEIN FUCOSYLATION IN VIVO USING FUCOSE ANALOGS SEATTLE GENETICS, INC. (US) 2013-05-23 US disclosed
US-20120183997-A1 METHODS AND COMPOSITIONS FOR MAKING ANTIBODIES AND ANTIBODY DERIVATIVES WITH REDUCED CORE FUCOSYLATION SEATTLE GENETICS, INC. (US) 2012-07-19 US disclosed
US-8163551-B2 Methods and compositions for making antibodies and antibody derivatives with reduced core fucosylation SEATTLE GENETICS, INC. (US) 2012-04-24 US disclosed
WO-2012019165-A2 METHODS OF INHIBITION OF PROTEIN FUCOSYLATION IN VIVO USING FUCOSE ANALOGS SEATTLE GENETICS, INC. (US) 2012-02-09 WO disclosed
US-20090317869-A1 METHODS AND COMPOSITIONS FOR MAKING ANTIBODIES AND ANTIBODY DERIVATIVES WITH REDUCED CORE FUCOSYLATION SEATTLE GENETICS, INC. (US) 2009-12-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140031536-A1 METHODS AND COMPOSITIONS FOR MAKING ANTIBODIES AND ANTIBODY DERIVATIVES WITH REDUCED CORE FUCOSYLATION FUT5, FUCA2, FCGR3B GBA1 226/4885ALDH1A1 3059/4885TSHR 1665/4885
US-20230055475-A1 METHODS AND COMPOSITIONS FOR MAKING ANTIBODIES AND ANTIBODY DERIVATIVES WITH REDUCED CORE FUCOSYLATION FUT5, FUCA2, FCGR3B GBA1 226/4885ALDH1A1 3059/4885TSHR 1665/4885
US-10443035-B2 Methods and compositions for making antibodies and antibody derivatives with reduced core fucosylation FUT5, FUCA2, FCGR3B GBA1 226/4885ALDH1A1 3059/4885TSHR 1665/4885
US-10342811-B2 Methods of inhibition of protein fucosylation in vivo using fucose analogs FUCA1, FUCA2, FUT4 GBA1 509/4885ALDH1A1 2623/4885TSHR 3062/4885
US-20200061091-A1 METHODS OF INHIBITION OF PROTEIN FUCOSYLATION IN VIVO USING FUCOSE ANALOGS FUCA1, FUCA2, FUT4 GBA1 509/4885ALDH1A1 2623/4885TSHR 3062/4885
US-11033561-B2 Methods of inhibition of protein fucosylation in vivo using fucose analogs FUCA1, FUCA2, FUT4 GBA1 509/4885ALDH1A1 2623/4885TSHR 3062/4885
US-20130129784-A1 METHODS OF INHIBITION OF PROTEIN FUCOSYLATION IN VIVO USING FUCOSE ANALOGS FUCA1, FUCA2, FUT4 GBA1 509/4885ALDH1A1 2623/4885TSHR 3062/4885
US-20190276796-A1 METHODS AND COMPOSITIONS FOR MAKING ANTIBODIES AND ANTIBODY DERIVATIVES WITH REDUCED CORE FUCOSYLATION FUT5, FUCA2, FCGR3B GBA1 226/4885ALDH1A1 3059/4885TSHR 1665/4885
US-11319526-B2 Methods and compositions for making antibodies and antibody derivatives with reduced core fucosylation FUT5, FUCA2, FCGR3B GBA1 226/4885ALDH1A1 3059/4885TSHR 1665/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.