SCHEMBL5704643

SCHEMBL5704643

N[C@@H](Cc1ccc(Cl)cc1)[C@H](O)C(F)(F)F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.52
SLC6A2 P23975 2/20 0.48
SLC6A3 Q01959 2/20 0.48
GAA P10253 2/20 0.46
PPARG P37231 2/20 0.38
PPARA Q07869 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ALDH1A1 P00352 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
HTR3E A5X5Y0 1/20 0.37
HTR3B O95264 1/20 0.37
HTR3A P46098 1/20 0.37
HTR3D Q70Z44 1/20 0.37
HTR3C Q8WXA8 1/20 0.37
CYP2D6 P10635 3/20 0.37
CYP1A2 P05177 2/20 0.37
CYP2C19 P33261 2/20 0.37
HTR2A P28223 1/20 0.36
HRH1 P35367 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9543643 0.84 ESR1 (0.37) ALDH1A1ESR1ESR2CYP3A4TAAR1
SCHEMBL5704618 0.84 ESR1 (0.53) SLC6A2ESR1ESR2TAAR1
SCHEMBL6556276 0.81 EPHX1 (0.48) SLC6A4SLC6A2SLC6A3CYP2D6TAAR1
SCHEMBL10622532 0.81 EPHX1 (0.48) SLC6A4SLC6A2SLC6A3CYP2D6TAAR1
Hydrochloric Acid SCHEMBL5711578 0.80 EPHX1 (0.47) SLC6A4SLC6A2SLC6A3CYP2D6TAAR1
Hydrochloric Acid SCHEMBL5381337 0.76 SLC6A4 (0.57) SLC6A4SLC6A2SLC6A3GAAPPARG
SCHEMBL5750538 0.74 CNR2 (0.49) SLC6A4SLC6A2SLC6A3PPARGPPARA
SCHEMBL10763436 0.74 SLC6A4 (0.67) SLC6A4SLC6A2SLC6A3PPARGPPARA
SCHEMBL6307263 0.73 HTR2A (0.54) CYP1A2HTR2AHTR2B
SCHEMBL5812524 0.73 SLC6A4 (0.53) SLC6A4SLC6A2SLC6A3PPARGPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1243576-B1 PROCESSES FOR PRODUCING (AMINOMETHYL)TRIFLUOROMETHYLCARBINOL DERIVATIVES DAINIPPON SUMITOMO PHARMA CO (JP) 2006-10-11 EP disclosed
US-6646150-B1 Reacting 1,3-oxazolidin-5-one derivative with trialkyl-(trifluoromethyl)silane; removing trialkylsilyl group; reductive decyclization DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 2003-11-11 US disclosed
EP-1243576-A1 PROCESSES FOR PRODUCING (AMINOMETHYL)TRIFLUOROCARBINOL DERIVATIVES Dainippon Pharmaceutical Co., Ltd. (JP) 2002-09-25 EP disclosed