SCHEMBL6556276

SCHEMBL6556276

NC(Cc1ccccc1)C(O)C(F)(F)F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.48
SLC15A1 P46059 1/20 0.47
CSNK1E P49674 1/20 0.46
ALPI P09923 1/20 0.46
PKM P14618 1/20 0.46
PTGS1 P23219 1/20 0.46
XIAP P98170 1/20 0.46
SLC7A5 Q01650 1/20 0.46
SLC6A2 P23975 2/20 0.45
TAAR1 Q96RJ0 2/20 0.45
MAOA P21397 1/20 0.45
SLC6A4 P31645 1/20 0.45
SLC6A3 Q01959 1/20 0.45
SIGMAR1 Q99720 1/20 0.45
CYP2A6 P11509 1/20 0.45
ADORA2A P29274 1/20 0.45
ADORA1 P30542 1/20 0.45
KDM4E B2RXH2 1/20 0.44
LMNA P02545 1/20 0.44
MAPK1 P28482 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10622532 1.00 EPHX1 (0.48) EPHX1SLC15A1CSNK1EALPIPKM
Hydrochloric Acid SCHEMBL5711578 0.98 EPHX1 (0.47) EPHX1SLC15A1CSNK1EALPIPKM
SCHEMBL27345872 0.84 SLC15A1 (0.44) EPHX1SLC15A1CSNK1EALPIPKM
SCHEMBL7275924 0.84 KDM4E (0.49) EPHX1SLC15A1CSNK1EALPIPKM
SCHEMBL7337442 0.84 KDM4E (0.49) EPHX1SLC15A1CSNK1EALPIPKM
SCHEMBL5704618 0.83 ESR1 (0.53) SLC7A5SLC6A2TAAR1
SCHEMBL9543643 0.83 ESR1 (0.37) CSNK1ETAAR1
SCHEMBL7412831 0.82 SLC15A1 (0.50) EPHX1SLC15A1CSNK1EALPIPKM
SCHEMBL7412834 0.82 SLC15A1 (0.50) EPHX1SLC15A1CSNK1EALPIPKM
SCHEMBL6351074 0.82 SLC15A1 (0.43) EPHX1SLC15A1CSNK1EALPIPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0826671-B1 HETEROCYCLIC AMIDE COMPOUNDS AND MEDICINAL USE OF THE SAME MITSUBISHI PHARMA CORP (JP) 2004-12-29 EP disclosed
EP-0721449-B1 INHIBITORS OF BETA-AMYLOID PROTEIN PRODUCTION MERRELL PHARMA INC (US) 2001-12-19 EP disclosed
US-5977074-A THERAPY FOR ALZHEIMER'S DISEASE MERRELL PHARMACEUTICALS, INC. (US) 1999-11-02 US disclosed
US-5948785-A USEFUL AS CHYMASE INHIBITORS AND CAN BE EFFECTIVE FOR THE PROPHYLAXIS AND TREATMENT OF VARIOUS DISEASES CAUSED BY CHYMASE, SUCH AS THOSE CAUSED BY ANGIOTENSIN II. THE GREEN CROSS CORPORATION (JP) 1999-09-07 US disclosed
EP-0826671-A1 HETEROCYCLIC AMIDE COMPOUNDS AND MEDICINAL USE OF THE SAME THE GREEN CROSS CORPORATION (JP) 1998-03-04 EP disclosed