SCHEMBL5706160

SCHEMBL5706160

CCOc1ccc(Br)c(C(=O)N[C@@H](Cc2ccc(-c3ccc(C#N)cc3OC)c(OC)c2)C(=O)O)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 6/20 0.48
ITGA4 P13612 5/20 0.48
ITGB2 P05107 1/20 0.46
ICAM1 P05362 1/20 0.46
ITGAL P20701 1/20 0.46
GPR34 Q9UPC5 1/20 0.42
PTPN1 P18031 1/20 0.41
GAA P10253 1/20 0.39
RAB9A P51151 1/20 0.39
SUCNR1 Q9BXA5 1/20 0.39
ITGB3 P05106 2/20 0.38
ITGAV P06756 1/20 0.38
ITGA5 P08648 1/20 0.38
PIN1 Q13526 1/20 0.38
PPARG P37231 1/20 0.37
CA2 P00918 1/20 0.37
ITGA2B P08514 1/20 0.37
EGLN1 Q9GZT9 1/20 0.37
PDCD1 Q15116 1/20 0.36
CD274 Q9NZQ7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5706239 0.93 GAA (0.45) ITGB1ITGA4ITGB2ICAM1ITGAL
SCHEMBL5706008 0.88 ITGB1 (0.48) ITGB1ITGA4ITGB2ICAM1ITGAL
SCHEMBL5706072 0.88 ITGB1 (0.45) ITGB1ITGA4ITGB2ICAM1ITGAL
SCHEMBL5706009 0.87 ITGB1 (0.45) ITGB1ITGA4ITGB2ICAM1ITGAL
SCHEMBL4648600 0.87 ITGB1 (0.52) ITGB1ITGA4ITGB2ICAM1ITGAL
SCHEMBL4649378 0.87 ITGB1 (0.52) ITGB1ITGA4ITGB2ICAM1ITGAL
Tetrahydrofuran SCHEMBL4648660 0.81 ITGB1 (0.47) ITGB1ITGA4ITGB2ICAM1ITGAL
SCHEMBL4649446 0.80 GAA (0.47) ITGB1ITGA4ITGB2ICAM1ITGAL
SCHEMBL4649444 0.80 GAA (0.47) ITGB1ITGA4ITGB2ICAM1ITGAL
SCHEMBL4649064 0.79 ITGA4 (0.59) ITGB1ITGA4ITGB2ICAM1ITGAL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1701933-A1 NOVEL COMPOUNDS TANABE SEIYAKU CO., LTD. (JP) 2006-09-20 EP disclosed
WO-2005061440-A1 NOVEL COMPOUNDS TANABE SEIYAKU CO., LTD. (JP) 2005-07-07 WO disclosed