SCHEMBL5706459

SCHEMBL5706459

OC(O)C(O)C(O)Cc1cnccn1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
DAO P14920 1/20 0.34
IDO1 P14902 1/20 0.33
VNN1 O95497 1/20 0.32
NAPRT Q6XQN6 1/20 0.31
HCAR2 Q8TDS4 1/20 0.31
HSP90AA1 P07900 1/20 0.31
CYP1A2 P05177 2/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
BAZ2B Q9UIF8 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL755982 0.81
SCHEMBL26085643 0.81 KDM4E (0.43) KDM4EALDH1A1SMN1; SMN2HDAC3HDAC1
SCHEMBL6966444 0.81 POLB (0.37) KDM4EALDH1A1SMN1; SMN2HDAC3HDAC1
SCHEMBL6965886 0.81 POLB (0.37) KDM4EALDH1A1SMN1; SMN2HDAC3HDAC1
SCHEMBL8105929 0.81 POLB (0.37) KDM4EALDH1A1SMN1; SMN2HDAC3HDAC1
SCHEMBL30638522 0.76 KDM4E (0.50) KDM4EALDH1A1SMN1; SMN2HDAC3HDAC1
SCHEMBL9474835 0.76 KDM4E (0.50) KDM4EALDH1A1SMN1; SMN2HDAC3HDAC1
SCHEMBL8351773 0.76 HSP90AA1 (0.38) KDM4EALDH1A1SMN1; SMN2HDAC3HDAC1
SCHEMBL28322787 0.74 DAO (0.38) KDM4EALDH1A1SMN1; SMN2HDAC3HDAC1
SCHEMBL10715444 0.73 KDM4E (0.40) KDM4EALDH1A1SMN1; SMN2HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1704862-A1 2,5-bis(tetrahydroxybutyl)pyrazines for the treatment of osteoarthritis and rheumatoid arthritis Rottapharm S.p.A. (IT) 2006-09-27 EP disclosed
CN-1148178-C Mixtures obtainable by isolation from seeds of Eugenia jambolana, their preparation, and use of these mixtures and certain components thereof as medicaments О 2004-05-05 CN disclosed
CN-1080566-C Mixtures obtainable by isolation from seeds of Eugenia jambolana, their preparation, and use of these mixtures and certain components thereof as medicaments INST OF MALGACHE DE RECHARCHES (MG) 2002-03-13 CN disclosed
CN-1325685-A Mixtures obtainable by isolation from seeds of Eugenia jambolana, their preparation, and use of these mixtures and certain components thereof as medicaments MADAGASCAR APPLIC INC (MG) 2001-12-12 CN disclosed
CN-1210469-A Mixtures obtainable by isolation from seeds of Eugenia jambolana, their preparation, and use of these mixtures and certain components thereof as medicaments INST MALGACHE RECH APPL (MG) 1999-03-10 CN disclosed