SCHEMBL8105929

SCHEMBL8105929

OCC(O)C(O)Cc1cnccn1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.37
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
DAO P14920 1/20 0.34
IDO1 P14902 1/20 0.33
VNN1 O95497 1/20 0.32
NAPRT Q6XQN6 1/20 0.31
HCAR2 Q8TDS4 1/20 0.31
HSP90AA1 P07900 1/20 0.31
CYP1A2 P05177 2/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
SYK P43405 1/20 0.31
BAZ2B Q9UIF8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6965886 1.00 POLB (0.37) POLBKDM4EALDH1A1SMN1; SMN2HDAC3
SCHEMBL6966444 1.00 POLB (0.37) POLBKDM4EALDH1A1SMN1; SMN2HDAC3
SCHEMBL28322787 0.82 DAO (0.38) POLBKDM4EALDH1A1SMN1; SMN2HDAC3
SCHEMBL26085643 0.81 KDM4E (0.43) POLBKDM4EALDH1A1SMN1; SMN2HDAC3
SCHEMBL5706459 0.81 KDM4E (0.36) POLBKDM4EALDH1A1SMN1; SMN2HDAC3
SCHEMBL7109077 0.78 LMNA (0.31)
SCHEMBL7109071 0.78 LMNA (0.31)
SCHEMBL7107159 0.78 LMNA (0.31)
SCHEMBL6094582 0.77 HSP90AA1 (0.35) POLBKDM4EALDH1A1SMN1; SMN2HDAC3
SCHEMBL20278973 0.77 HSP90AA1 (0.35) POLBKDM4EALDH1A1SMN1; SMN2HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1264368-A Polyhydroxybutylpyrazines, process for their preparation and medicaments containing them RHONE POULENC RORER SA (FR) 2000-08-23 CN disclosed
EP-1001943-A1 POLYHYDROXYALKYLPYRAZINE DERIVATIVES, PREPARATION AND MEDICINES CONTAINING THEM Aventis Pharma S.A. (FR) 2000-05-24 EP disclosed
US-5972342-A ANTIDIABETIC AGENTS RHONE-POULENC RORER S.A. (FR) 1999-10-26 US disclosed
WO-1999003843-A1 POLYHYDROXYALKYLPYRAZINE DERIVATIVES, PREPARATION AND MEDICINES CONTAINING THEM RHONE-POULENC RORER S.A. (FR) 1999-01-28 WO disclosed