SCHEMBL5709394

SCHEMBL5709394

O=C(O)CC(c1ccc(Cl)cc1)c1ccc(F)c(F)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 2/20 0.52
GABBR2 O75899 3/20 0.50
GABBR1 Q9UBS5 3/20 0.50
CYP2C9 P11712 3/20 0.50
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
LMNA P02545 2/20 0.50
CYP2D6 P10635 2/20 0.50
CYP2C19 P33261 2/20 0.50
CYP3A4 P08684 1/20 0.50
ADORA3 P0DMS8 1/20 0.50
NFKB1 P19838 1/20 0.50
DRD3 P35462 1/20 0.50
BLM P54132 1/20 0.50
CYP1A2 P05177 1/20 0.50
THRB P10828 1/20 0.50
TSHR P16473 1/20 0.50
HSD17B10 Q99714 1/20 0.46
FFAR1 O14842 3/20 0.43
PPARG P37231 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5709322 0.91 KEAP1 (0.46) KEAP1GABBR2GABBR1CYP2C9MEN1
SCHEMBL3520190 0.86 GABBR2 (0.63) KEAP1GABBR2GABBR1CYP2C9MEN1
Hydrochloric Acid SCHEMBL11527826 0.84 GABBR2 (0.61) KEAP1GABBR2GABBR1CYP2C9MEN1
SCHEMBL22089315 0.83 GABBR2 (0.50) KEAP1GABBR2GABBR1CYP2C9MEN1
SCHEMBL15872203 0.81 GAA (0.48) KEAP1CYP2C9CYP2C19FFAR1CES2
SCHEMBL15872205 0.81 GAA (0.48) KEAP1CYP2C9CYP2C19FFAR1CES2
SCHEMBL6002264 0.80 GABBR2 (0.58) KEAP1GABBR2GABBR1CYP2C9MEN1
SCHEMBL15614165 0.80 GABBR2 (0.58) KEAP1GABBR2GABBR1CYP2C9MEN1
SCHEMBL7809416 0.79 GABBR2 (0.47) GABBR2GABBR1CYP2C9MEN1KMT2A
SCHEMBL3030480 0.78 FFAR1 (0.51) KEAP1KMT2AFFAR1PPARGPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1727785-A1 PHENYL INDAN DERIVATIVES H.Lundbeck A/S (DK) 2006-12-06 EP disclosed
WO-2005087708-A1 PHENYL INDAN DERIVATIVES H. LUNDBECK A/S (DK) 2005-09-22 WO disclosed