SCHEMBL5709778

SCHEMBL5709778

O=C(Cc1ccccc1)C(F)(F)F.O=C(Cc1ccccc1)C(F)(F)F

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CES1 P23141 7/20 1.00
FAAH O00519 3/20 0.56
CES2 O00748 1/20 0.56
AKR1B1 P15121 1/20 0.56
CPA1 P15085 1/20 0.55
PTPN1 P18031 1/20 0.50
PAM P19021 1/20 0.48
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
FNTA P49354 1/20 0.47
FNTB P49356 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1042453 1.00 CES1 (1.00) CES1FAAHCES2AKR1B1CPA1
SCHEMBL583920 0.88 CES1 (0.78) CES1FAAHMEN1KMT2AHDAC8
SCHEMBL4753311 0.84 CES1 (0.71) CES1FAAHCES2AKR1B1CPA1
SCHEMBL2381708 0.83 CES1 (0.69) CES1HDAC6
SCHEMBL16405134 0.83 CES1 (0.70) CES1FAAHCES2AKR1B1CPA1
SCHEMBL13498524 0.83 CES1 (0.70) CES1FAAHCES2AKR1B1CPA1
SCHEMBL9314779 0.83 CES1 (0.70) CES1FAAHCES2AKR1B1CPA1
SCHEMBL10433444 0.83 CES1 (0.70) CES1FAAHCES2AKR1B1CPA1
Phenylacetic Acid SCHEMBL27489228 0.80 AKR1B1 (0.74) CES1CES2AKR1B1CPA1PAM
SCHEMBL10431529 0.80 CES1 (0.67) CES1FNTAFNTB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1732531-A2 AMINES AND AMIDES FOR THE TREATMENT OF DISEASES LA JOLLA PHARMACEUTICAL COMPANY (US) 2006-12-20 EP disclosed
WO-2005082343-A2 AMINES AND AMIDES FOR THE TREATMENT OF DISEASES LA JOLLA PHARMACEUTICAL COMPANY (US) 2005-09-09 WO disclosed