SCHEMBL583920

SCHEMBL583920

O=C(Cc1ccc(-c2ccccc2)cc1)C(F)(F)F

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 4/20 0.78
LMNA P02545 2/20 0.62
ABCC4 O15439 1/20 0.62
GAA P10253 1/20 0.62
TSHR P16473 1/20 0.62
PTGS1 P23219 1/20 0.62
HTT P42858 1/20 0.62
KMT2A Q03164 3/20 0.51
MEN1 O00255 2/20 0.51
HDAC1 Q13547 4/20 0.50
HDAC2 Q92769 4/20 0.50
HDAC3 O15379 3/20 0.50
HDAC4 P56524 3/20 0.50
HDAC7 Q8WUI4 3/20 0.50
HDAC10 Q969S8 3/20 0.50
HDAC11 Q96DB2 3/20 0.50
HDAC8 Q9BY41 3/20 0.50
HDAC6 Q9UBN7 3/20 0.50
HDAC9 Q9UKV0 3/20 0.50
HDAC5 Q9UQL6 3/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1042453 0.88 CES1 (1.00) CES1KMT2AMEN1HDAC8HDAC6
SCHEMBL5709778 0.88 CES1 (1.00) CES1KMT2AMEN1HDAC8HDAC6
SCHEMBL583919 0.81 FFAR1 (0.65) CES1LMNAABCC4GAATSHR
SCHEMBL12895712 0.81 LMNA (0.62) CES1LMNAABCC4GAATSHR
SCHEMBL10431529 0.78 CES1 (0.67) CES1LMNA
SCHEMBL28262050 0.77 CES1 (0.56) CES1LMNAABCC4GAATSHR
Felbinac SCHEMBL26084 0.77 LMNA (1.00) LMNAABCC4GAATSHRPTGS1
SCHEMBL11879591 0.77 LMNA (0.75) CES1LMNAABCC4GAATSHR
SCHEMBL2381708 0.76 CES1 (0.69) CES1LMNAPTGS1HDAC6FFAR1
SCHEMBL17073597 0.76 CES1 (0.64) CES1LMNAGAAKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118108572-A Synthesis method of alkyl trifluoromethyl compounds 合肥工业大学 2024-05-31 CN disclosed
EP-2417216-A2 MODIFICATION OF LAYERED SILICATES FOR LUMINESCENCE ACTIVATION Inbio Prof. Jürgen Büddefeld Dr. Peter Klauth Prof. Manfred Rietz Gbr (DE) 2012-02-15 EP disclosed
WO-2010115503-A2 MODIFICATION OF LAYERED SILICATES FOR LUMINESCENCE ACTIVATION INBIO PROF. JÜRGEN BÜDDEFELD DR. PETER KLAUTH PROF. MANFRED RIETZ GBR (DE) 2010-10-14 WO disclosed