SCHEMBL5710778

SCHEMBL5710778

O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTRB1 P17538 1/20 0.74
KMT2A Q03164 2/20 0.60
NPSR1 Q6W5P4 1/20 0.58
TSHR P16473 3/20 0.57
L3MBTL1 Q9Y468 1/20 0.57
KDM4E B2RXH2 1/20 0.57
LMNA P02545 1/20 0.57
GFER P55789 1/20 0.56
HSD17B10 Q99714 1/20 0.56
ACE P12821 1/20 0.56
PREP P48147 2/20 0.56
ALDH1A1 P00352 2/20 0.56
KDM1A O60341 1/20 0.56
RCOR1 Q9UKL0 1/20 0.56
CTSL P07711 1/20 0.55
CTSK P43235 1/20 0.55
CYP3A4 P08684 1/20 0.55
MAPT P10636 1/20 0.55
CYP2C9 P11712 1/20 0.55
RAB9A P51151 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30439776 1.00 CTRB1 (0.74) CTRB1KMT2ANPSR1TSHRL3MBTL1
SCHEMBL7702739 0.96 CTRB1 (0.69) CTRB1KMT2ANPSR1TSHRL3MBTL1
SCHEMBL11243030 0.93 CTRB1 (0.66) CTRB1KMT2ANPSR1TSHRL3MBTL1
SCHEMBL6367959 0.90 CTRB1 (0.62) CTRB1NPSR1ALDH1A1MAPT
SCHEMBL24513611 0.89 CTRB1 (0.64) CTRB1KMT2ANPSR1TSHRL3MBTL1
SCHEMBL11167627 0.89 CTRB1 (0.64) CTRB1KMT2ANPSR1TSHRL3MBTL1
SCHEMBL11167632 0.89 CTRB1 (0.64) CTRB1KMT2ANPSR1TSHRL3MBTL1
SCHEMBL11450738 0.89 CTRB1 (0.64) CTRB1KMT2ANPSR1TSHRL3MBTL1
SCHEMBL7106091 0.89 CTRB1 (0.64) CTRB1KMT2ANPSR1TSHRL3MBTL1
SCHEMBL2557292 0.89 CTRB1 (0.64) CTRB1KMT2ANPSR1TSHRL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119371478-A Method for synthesizing amide and/or polypeptide by taking transient protection amino acid as ammonia component 广州医科大学 2025-01-28 CN disclosed
WO-2025015659-A1 METHOD FOR SYNTHESIZING AMIDE AND/OR POLYPEPTIDE BY TAKING TRANSIENTLY PROTECTED AMINO ACID AS AMMONIA COMPONENT 广州医科大学 2025-01-23 WO disclosed
EP-4135660-A1 COMPOSITIONS AND METHODS TO REDUCE THE INFECTIVITY OF A VIRUS Atossa Therapeutics, Inc. (US) 2023-02-22 EP disclosed
WO-2021211808-A1 COMPOSITIONS AND METHODS TO REDUCE THE INFECTIVITY OF A VIRUS ATOSSA THERAPEUTICS, INC. (US) 2021-10-21 WO disclosed
EP-1715885-A2 COMPOSITIONS AND METHODS FOR ENHANCED MUCOSAL DELIVERY OF Y2 RECEPTOR-BINDING PEPTIDES AND METHODS FOR TREATING AND PREVENTING OBESITY Nastech Pharmaceutical Company Inc. (US) 2006-11-02 EP disclosed
EP-1696960-A1 INTRANASAL ADMINISTRATION OF GLUCOSE-REGULATING PEPTIDES Nastech Pharmaceutical Company Inc. (US) 2006-09-06 EP disclosed
EP-1581245-A2 COMPOSITIONS AND METHODS FOR ENHANCED MUCOSAL DELIVERY OF Y2 RECEPTOR-BINDING PEPTIDES AND METHODS FOR TREATING AND PREVENTING OBESITY Nastech Pharmaceutical Company Inc. (US) 2005-10-05 EP disclosed
WO-2005080433-A2 COMPOSITIONS AND METHODS FOR ENHANCED MUCOSAL DELIVERY OF Y2 RECEPTOR-BINDING PEPTIDES AND METHODS FOR TREATING AND PREVENTING OBESITY NASTECH PHARMACEUTICAL COMPANY INC. (US) 2005-09-01 WO disclosed
WO-2005065714-A1 INTRANASAL ADMINISTRATION OF GLUCOSE-REGULATING PEPTIDES NASTECH PHARMACEUTICAL COMPANY INC. (US) 2005-07-21 WO disclosed
WO-2004056314-A2 COMPOSITIONS AND METHODS FOR ENHANCED MUCOSAL DELIVERY OF Y2 RECEPTOR-BINDING PEPTIDES AND METHODS FOR TREATING AND PREVENTING OBESITY NASTECH PHARMACEUTICAL COMPANY INC. (US) 2004-07-08 WO disclosed
US-6066482-A AMINO ACID SEQUENCES; FOR PRODUCING SUGAR POLYESTERS WITH PEST REPELLENT PROPERTIES USED IN AGRICULTURE, EMULSIFICATION PROPERTIES USED IN FOOD AND COSMETIC INDUSTRIES, AND EMOLLIENT PROPERTIES USED IN COSMETICS CORNELL RESEARCH FOUNDATION, INC. (US) 2000-05-23 US disclosed
EP-0909326-A1 ACYLTRANSFERASE AND GENE ENCODING ACYLTRANSFERASE CORNELL RESEARCH FOUNDATION, INC. (US) 1999-04-21 EP disclosed
US-5756328-A PURE ENZYME WHICH CATALYZES TRANSFER OF ACYL SUBSTITUENTS TO PRODUCE SUGAR ESTERS OR SUGAR POLYESTERS, HAVING SPECIFIED AMINO ACID SEQUENCE CORNELL RESEARCH FOUNDATION, INC. (US) 1998-05-26 US disclosed
WO-1997048811-A1 ACYLTRANSFERASE AND GENE ENCODING ACYLTRANSFERASE CORNELL RESEARCH FOUNDATION, INC. (US) 1997-12-24 WO disclosed
US-4350628-A OXIDATIVE DEHYDROGENATION WITH A BENZOQUINONE RESEARCH CORPORATION (US) 1982-09-21 US disclosed
US-4308202-A Prolylphenylalanylarginine derivatives, process for producing same and method for measuring activity of enzymes using same TORII & CO., LTD. (JP) 1981-12-29 US disclosed
US-4283328-A TREATING AN N-BLOCKED AMINO ACID RESIDUE WITH A TETRAMETHYL GUANIDINIUM SALT OF A PEPTIDE CHAIN RESEARCH CORPORATION (US) 1981-08-11 US disclosed
US-4261884-A DESIRABLE BIOLOGICAL PROPERTIES AND STABILITY TO ENZYME CLEAVAGE RESEARCH CORPORATION (US) 1981-04-14 US disclosed
EP-0010830-A2 Dehydropeptides Research Corporation (US) 1980-05-14 EP disclosed