SCHEMBL11243030

SCHEMBL11243030

O=C(O)[C@H](Cc1ccc(OCc2ccccc2)cc1)NC(=O)[C@@H]1CCCN1C(=O)OCc1ccccc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTRB1 P17538 1/20 0.66
KDM4E B2RXH2 1/20 0.61
LMNA P02545 1/20 0.61
ACE P12821 3/20 0.58
HDAC1 Q13547 1/20 0.57
NPSR1 Q6W5P4 1/20 0.55
ALDH1A1 P00352 1/20 0.54
TSHR P16473 2/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
KMT2A Q03164 1/20 0.54
ITGB3 P05106 1/20 0.54
ITGA2B P08514 1/20 0.54
TP53 P04637 1/20 0.54
YAP1 P46937 2/20 0.53
CYP3A4 P08684 1/20 0.51
MAPT P10636 1/20 0.51
CYP2C9 P11712 1/20 0.51
RAB9A P51151 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
PPARG P37231 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30439776 0.93 CTRB1 (0.74) CTRB1KDM4ELMNAACENPSR1
SCHEMBL5710778 0.93 CTRB1 (0.74) CTRB1KDM4ELMNAACENPSR1
SCHEMBL7702739 0.91 CTRB1 (0.69) CTRB1KDM4ELMNAACENPSR1
SCHEMBL6367959 0.88 CTRB1 (0.62) CTRB1NPSR1ALDH1A1MAPT
SCHEMBL21429800 0.86 YAP1 (0.59) CTRB1KDM4ELMNAACENPSR1
SCHEMBL19639223 0.84 CTRB1 (0.67) CTRB1KDM4ELMNAACENPSR1
SCHEMBL11434855 0.83 CTRB1 (0.60) CTRB1KDM4ELMNANPSR1ALDH1A1
SCHEMBL11434851 0.83 CTRB1 (0.60) CTRB1KDM4ELMNANPSR1ALDH1A1
SCHEMBL24513611 0.82 CTRB1 (0.64) CTRB1KDM4ELMNANPSR1ALDH1A1
SCHEMBL11167627 0.82 CTRB1 (0.64) CTRB1KDM4ELMNANPSR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4350628-A OXIDATIVE DEHYDROGENATION WITH A BENZOQUINONE RESEARCH CORPORATION (US) 1982-09-21 US disclosed
US-4283328-A TREATING AN N-BLOCKED AMINO ACID RESIDUE WITH A TETRAMETHYL GUANIDINIUM SALT OF A PEPTIDE CHAIN RESEARCH CORPORATION (US) 1981-08-11 US disclosed
US-4261884-A DESIRABLE BIOLOGICAL PROPERTIES AND STABILITY TO ENZYME CLEAVAGE RESEARCH CORPORATION (US) 1981-04-14 US disclosed