SCHEMBL5717019

SCHEMBL5717019

CCOC(=O)C1CCCCN1S(=O)(=O)c1ccc(Br)cc1C

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 5/20 0.60
HCRTR2 O43614 5/20 0.60
FKBP1A P62942 7/20 0.54
MMP1 P03956 1/20 0.49
MMP2 P08253 1/20 0.49
MMP3 P08254 1/20 0.49
MMP7 P09237 1/20 0.49
MMP13 P45452 1/20 0.49
ALDH1A1 P00352 3/20 0.47
TSHR P16473 2/20 0.47
KDM4E B2RXH2 2/20 0.47
KMT2A Q03164 2/20 0.45
MEN1 O00255 1/20 0.45
MAPK1 P28482 1/20 0.45
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5717109 0.86 KDM4E (0.51) HCRTR1HCRTR2FKBP1AALDH1A1TSHR
SCHEMBL5717089 0.85 ALDH1A1 (0.58) HCRTR1HCRTR2FKBP1AALDH1A1TSHR
SCHEMBL5717045 0.84 FKBP1A (0.64) HCRTR1HCRTR2FKBP1AMMP1MMP3
SCHEMBL2704252 0.81 HCRTR1 (0.70) HCRTR1HCRTR2MMP1MMP2MMP3
SCHEMBL2704254 0.81 HCRTR1 (0.70) HCRTR1HCRTR2MMP1MMP2MMP3
SCHEMBL5717267 0.80 ALDH1A1 (0.55) HCRTR1HCRTR2FKBP1AALDH1A1TSHR
SCHEMBL19975403 0.76 HCRTR1 (0.50) HCRTR1HCRTR2FKBP1AMMP1MMP2
SCHEMBL5717026 0.76 FKBP1A (0.50) HCRTR1HCRTR2FKBP1AALDH1A1TSHR
SCHEMBL5717002 0.76 HCRTR1 (0.62) HCRTR1HCRTR2FKBP1AALDH1A1TSHR
SCHEMBL19975023 0.74 FKBP1A (0.48) HCRTR1HCRTR2FKBP1AMMP1MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1664010-A1 SULFONAMIDES ANTAGONISING N-TYPE CALCIUM CHANNELS Vernalis (R&D) Limited (GB) 2006-06-07 EP disclosed
WO-2005068448-A1 SULFONAMIDES ANTAGONISING N-TYPE CALCIUM CHANNELS IONIX PHARMACEUTICALS LIMITED (GB) 2005-07-28 WO disclosed