SCHEMBL5718014

SCHEMBL5718014

NCC(=O)Nc1ccccc1C(=O)[C@H]1CCCC[C@H]1c1ccc(CN(C(=O)NCCO)c2ccccc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTB4R2 Q9NPC1 4/20 0.40
KDM4E B2RXH2 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
GCGR P47871 5/20 0.33
GIPR P48546 3/20 0.33
KCNQ3 O43525 1/20 0.32
KCNQ2 O43526 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
ADRA2C P18825 1/20 0.32
PDK1 Q15118 1/20 0.32
STAT3 P40763 1/20 0.32
CHRM2 P08172 1/20 0.32
CHRM1 P11229 1/20 0.32
CHRM3 P20309 1/20 0.32
ITGA4 P13612 1/20 0.32
ITGB7 P26010 1/20 0.32
ABCC1 P33527 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5718010 0.87 LTB4R2 (0.34) LTB4R2KDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL5718017 0.79 LTB4R2 (0.40) LTB4R2GCGRGIPRKCNQ3KCNQ2
SCHEMBL5864496 0.71 PPARG (0.44)
SCHEMBL5864456 0.68 CYP2D6 (0.44) CHRM1
SCHEMBL5718013 0.66 KCNQ3 (0.37) LTB4R2GCGRGIPRKCNQ3KCNQ2
SCHEMBL5864492 0.65 KDM4E (0.38) KDM4EALDH1A1
SCHEMBL5718068 0.64 ATM (0.40) LTB4R2KCNQ3KCNQ2SLC6A2SLC6A4
SCHEMBL6733188 0.64 ALDH1A1 (0.40) LTB4R2SMN1; SMN2KCNQ3KCNQ2SLC6A2
SCHEMBL6737598 0.62 SLC6A2 (0.45) KCNQ3KCNQ2SLC6A2SLC6A4
SCHEMBL5718155 0.61 ALDH1A1 (0.42) LTB4R2KDM4ECHRM2CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1318977-B1 SUBSTITUTED PHENYLCYCLOHEXANE CARBOXYLIC ACID AMIDES AND THE USE THEREOF BAYER HEALTHCARE AG (DE) 2006-12-06 EP claimed
EP-1318977-B1 SUBSTITUTED PHENYLCYCLOHEXANE CARBOXYLIC ACID AMIDES AND THE USE THEREOF BAYER HEALTHCARE AG (DE) 2006-12-06 EP disclosed