SCHEMBL5718487

SCHEMBL5718487

CN(CC(=O)N(c1ccccc1)c1ccccc1)C1CCN(Cc2ccccc2)C1

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 4/20 0.57
SIGMAR1 Q99720 4/20 0.57
CHRM2 P08172 8/20 0.55
CHRM3 P20309 8/20 0.55
CHRM4 P08173 1/20 0.54
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
LTA4H P09960 1/20 0.52
KCNH2 Q12809 1/20 0.48
HTR2A P28223 2/20 0.48
HTR2C P28335 2/20 0.48
HTR2B P41595 2/20 0.48
DRD2 P14416 1/20 0.48
CCR5 P51681 1/20 0.47
ACHE P22303 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4464056 1.00 OPRM1 (0.57) OPRM1SIGMAR1CHRM2CHRM3CHRM4
SCHEMBL6312702 0.86 CHRM4 (0.59) OPRM1SIGMAR1CHRM2CHRM3CHRM4
SCHEMBL8283548 0.86 CHRM4 (0.49) OPRM1SIGMAR1CHRM2CHRM3CHRM4
SCHEMBL4463836 0.81 OPRM1 (0.57) OPRM1SIGMAR1CHRM2CHRM3CHRM4
SCHEMBL4463840 0.81 OPRM1 (0.57) OPRM1SIGMAR1CHRM2CHRM3CHRM4
SCHEMBL3817982 0.78 OPRM1 (0.59) OPRM1SIGMAR1CHRM2CHRM3CHRM4
SCHEMBL1220330 0.78 OPRM1 (0.59) OPRM1SIGMAR1CHRM2CHRM3CHRM4
SCHEMBL7013887 0.78 SIGMAR1 (0.60) OPRM1SIGMAR1CHRM2CHRM3CHRM4
SCHEMBL11577007 0.78 OPRM1 (0.86) OPRM1SIGMAR1CHRM2CHRM3MEN1
SCHEMBL4891859 0.78 CHRM3 (0.57) OPRM1SIGMAR1CHRM2CHRM3CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1718633-A1 N-TYPE CALCIUM CHANNEL BLOCKERS Neuromed Pharmaceuticals, Ltd. (CA) 2006-11-08 EP disclosed
WO-2005070919-A1 N-TYPE CALCIUM CHANNEL BLOCKERS NEUROMED PHARMACEUTICALS LTD. (CA) 2005-08-04 WO disclosed