SCHEMBL5718890

SCHEMBL5718890

CC#CCn1c(N2CCN(C(=O)O)CC2)nc2c1c(=O)[nH]c(=O)n2CCOCC

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.54
RAB9A P51151 1/20 0.54
MAPT P10636 1/20 0.49
ALOX15 P16050 1/20 0.49
ALDH1A1 P00352 5/20 0.43
GAA P10253 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
TP53 P04637 1/20 0.42
DPP4 P27487 2/20 0.41
HPGD P15428 1/20 0.41
POLB P06746 1/20 0.41
MAPK1 P28482 2/20 0.41
HSD17B10 Q99714 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
LMNA P02545 1/20 0.40
TSHR P16473 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5719333 0.89 NPC1 (0.48) NPC1RAB9AMAPTALOX15ALDH1A1
SCHEMBL5719595 0.87 DPP4 (0.56) NPC1RAB9AMAPTALOX15ALDH1A1
Trifluoroacetic Acid SCHEMBL5719362 0.85 DPP4 (0.49) NPC1RAB9AMAPTALOX15ALDH1A1
SCHEMBL5776712 0.81 GAA (0.39) ALDH1A1GAAL3MBTL1TP53DPP4
SCHEMBL6386721 0.75 DPP4 (0.47) DPP4
SCHEMBL5718802 0.75 GAA (0.52) ALDH1A1GAAL3MBTL1TP53DPP4
SCHEMBL5719799 0.74 DPP4 (0.59) ALDH1A1DPP4SMN1; SMN2
Trifluoroacetic Acid SCHEMBL5718899 0.73 DPP4 (0.57) ALDH1A1DPP4SMN1; SMN2
SCHEMBL5719154 0.73 ALDH1A1 (0.41) ALDH1A1GAAL3MBTL1TP53DPP4
SCHEMBL5719433 0.73 DPP4 (0.74) ALDH1A1DPP4SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1338595-B1 Xanthine derivatives as DPP-IV inhibitors EISAI CO LTD (JP) 2006-05-03 EP disclosed