SCHEMBL5720167

SCHEMBL5720167

O=C1[N]c2cc(C3CCN(C4CCN(Cc5sccc5Cl)CC4)CC3)ccc2N1

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TLR9 Q9NR96 7/20 0.35
TLR7 Q9NYK1 7/20 0.35
DRD2 P14416 6/20 0.34
DRD4 P21917 5/20 0.34
DRD3 P35462 3/20 0.34
TLR8 Q9NR97 4/20 0.33
CHRM1 P11229 3/20 0.33
TRPV6 Q9H1D0 4/20 0.33
PARP1 P09874 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5720129 0.89 TLR9 (0.35) TLR9TLR7DRD2DRD4DRD3
SCHEMBL5720269 0.89 DRD2 (0.39) TLR9TLR7DRD2DRD4DRD3
SCHEMBL5720110 0.84 TLR9 (0.40) TLR9TLR7DRD2DRD4DRD3
SCHEMBL5719999 0.83 CHRM2 (0.45) TLR9TLR7DRD2DRD4DRD3
SCHEMBL5720185 0.81 DRD2 (0.34) TLR9TLR7DRD2DRD4DRD3
SCHEMBL5720295 0.81 ALDH1A1 (0.36) CHRM1
SCHEMBL5720128 0.80 TLR7 (0.44) TLR9TLR7DRD2DRD4DRD3
SCHEMBL5720388 0.79 DRD2 (0.40) TLR9TLR7DRD2DRD4DRD3
SCHEMBL5720132 0.78 TRPV6 (0.41) TLR9TLR7DRD2DRD4DRD3
SCHEMBL5720125 0.78 CHRM1 (0.41) TLR9TLR7DRD2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1515722-A4 OPHTHALMIC COMPOSITIONS FOR TREATING OCULAR HYPERTENSION MERCK & CO INC (US) 2006-06-21 EP claimed
EP-1515722-A2 OPHTHALMIC COMPOSITIONS FOR TREATING OCULAR HYPERTENSION Merck & Co., Inc. (US) 2005-03-23 EP claimed
WO-2003105781-A2 OPHTHALMIC COMPOSITIONS FOR TREATING OCULAR HYPERTENSION MERCK & CO., INC. (US) 2003-12-24 WO claimed
EP-1515722-A4 OPHTHALMIC COMPOSITIONS FOR TREATING OCULAR HYPERTENSION MERCK & CO INC (US) 2006-06-21 EP disclosed
EP-1515722-A2 OPHTHALMIC COMPOSITIONS FOR TREATING OCULAR HYPERTENSION Merck & Co., Inc. (US) 2005-03-23 EP disclosed
WO-2003105781-A2 OPHTHALMIC COMPOSITIONS FOR TREATING OCULAR HYPERTENSION MERCK & CO., INC. (US) 2003-12-24 WO disclosed