SCHEMBL5723026

SCHEMBL5723026

Cc1ccc(S(=O)(=O)NNC(=O)[C@@H]2C[C@@H](S)CN2S(=O)(=O)c2ccc(C(F)(F)F)cc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ECE1 P42892 2/20 0.48
MME P08473 1/20 0.48
ACE P12821 1/20 0.48
ALDH1A1 P00352 3/20 0.47
POLB P06746 2/20 0.44
HTT P42858 1/20 0.44
MMP1 P03956 1/20 0.44
ADAM17 P78536 1/20 0.44
GAA P10253 2/20 0.42
KMT2A Q03164 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
MMP8 P22894 2/20 0.42
MMP3 P08254 1/20 0.42
TRPA1 O75762 2/20 0.42
LMNA P02545 1/20 0.41
CAPN1 P07384 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5724342 0.92 ALDH1A1 (0.55) ECE1MMEACEALDH1A1POLB
SCHEMBL5723387 0.90 MME (0.51) ECE1MMEACEALDH1A1POLB
SCHEMBL5722907 0.89 GAA (0.53) ECE1MMEACEALDH1A1POLB
SCHEMBL5723144 0.88 ECE1 (0.55) ECE1MMEACEALDH1A1POLB
SCHEMBL5723356 0.88 ALDH1A1 (0.51) ECE1MMEACEALDH1A1POLB
SCHEMBL5723752 0.87 ALDH1A1 (0.59) ECE1MMEACEALDH1A1POLB
SCHEMBL5723111 0.85 ALDH1A1 (0.49) ECE1MMEACEALDH1A1POLB
SCHEMBL5723189 0.85 MMP9 (0.54) ECE1MMEACEALDH1A1POLB
SCHEMBL5723156 0.85 MME (0.53) ECE1MMEACEALDH1A1POLB
SCHEMBL5722877 0.85 MMP1 (0.56) ECE1MMEACEALDH1A1MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1317428-B1 PYRROLIDINE-2-CARBOXYLIC ACID HYDRAZIDE DERIVATIVES FOR USE AS METALLOPROTEASE INHIBITORS HOFFMANN LA ROCHE (CH) 2006-04-19 EP disclosed