SCHEMBL5723201

SCHEMBL5723201

COCCOCCOc1nc(Cl)ncc1C#N

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 3/20 0.49
CSNK1A1 P48729 1/20 0.44
CLK4 Q9HAZ1 1/20 0.44
SRC P12931 6/20 0.37
USP8 P40818 1/20 0.36
AR P10275 1/20 0.36
SQOR Q9Y6N5 1/20 0.34
TSHR P16473 1/20 0.34
KCNJ5 P48544 3/20 0.34
KCNJ3 P48549 3/20 0.34
GAA P10253 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
FGFR4 P22455 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5723859 0.96 PIN1 (0.52) PIN1CSNK1A1CLK4SRCUSP8
SCHEMBL5723448 0.81 PIN1 (0.52) PIN1CSNK1A1CLK4SRCAR
SCHEMBL20101542 0.79 PIN1 (0.51) PIN1CSNK1A1CLK4GAAL3MBTL1
SCHEMBL5723588 0.79 PIN1 (0.56) PIN1CSNK1A1CLK4SRCSQOR
SCHEMBL2527306 0.78 PIN1 (0.59) PIN1CSNK1A1CLK4GAAL3MBTL1
SCHEMBL5723434 0.77 PIN1 (0.51) PIN1CSNK1A1CLK4GAAL3MBTL1
SCHEMBL22895389 0.75 TSHR (0.41) PIN1USP8TSHRKCNJ5KCNJ3
SCHEMBL5723482 0.74 PIN1 (0.51) PIN1CSNK1A1CLK4GAAL3MBTL1
SCHEMBL5723463 0.73 PIN1 (0.54) PIN1CSNK1A1CLK4GAAL3MBTL1
SCHEMBL23835201 0.72 SRC (0.38) PIN1CSNK1A1CLK4SRCUSP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1406876-B1 2-ANILINO-PYRIMIDINE DERIVATIVES AS CYCLIN DEPENDENT KINASE INHIBITORS ASTRAZENECA AB (SE) 2006-12-27 EP disclosed