SCHEMBL5723482

SCHEMBL5723482

CC#CCOc1nc(Cl)ncc1C#N

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 3/20 0.51
CSNK1A1 P48729 1/20 0.46
CLK4 Q9HAZ1 1/20 0.46
GAA P10253 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
KDM4E B2RXH2 1/20 0.34
MAPT P10636 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
CHRM3 P20309 1/20 0.32
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5723463 0.81 PIN1 (0.54) PIN1CSNK1A1CLK4GAAL3MBTL1
SCHEMBL5723588 0.81 PIN1 (0.56) PIN1CSNK1A1CLK4GAAL3MBTL1
SCHEMBL2527306 0.77 PIN1 (0.59) PIN1CSNK1A1CLK4GAAL3MBTL1
SCHEMBL5723448 0.77 PIN1 (0.52) PIN1CSNK1A1CLK4GAAL3MBTL1
SCHEMBL5723859 0.77 PIN1 (0.52) PIN1CSNK1A1CLK4GAAL3MBTL1
SCHEMBL20101542 0.76 PIN1 (0.51) PIN1CSNK1A1CLK4GAAL3MBTL1
SCHEMBL5723291 0.74 PIN1 (0.52) PIN1CSNK1A1CLK4
SCHEMBL15831947 0.74 HDAC1 (0.41) GAAL3MBTL1KDM4EMAPTTDP1
SCHEMBL5723201 0.74 PIN1 (0.49) PIN1CSNK1A1CLK4GAAL3MBTL1
SCHEMBL5723781 0.73 PIN1 (0.55) PIN1CSNK1A1CLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1406876-B1 2-ANILINO-PYRIMIDINE DERIVATIVES AS CYCLIN DEPENDENT KINASE INHIBITORS ASTRAZENECA AB (SE) 2006-12-27 EP disclosed
US-6939872-B2 2-anilino-pyrimidine derivatives as cyclin dependent kinase inhibitors ASTRAZENECA AB (SE) 2005-09-06 US disclosed