SCHEMBL5723402

SCHEMBL5723402

CS(=O)(=O)c1ccc(S(=O)(=O)NNC(=O)[C@@H]2C[C@@H](S)CN2S(=O)(=O)c2ccc3ccccc3c2)cc1

nearest known ligand 0.61

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ECE1 P42892 3/20 0.61
MME P08473 2/20 0.61
ACE P12821 2/20 0.61
KAT6A Q92794 11/20 0.44
EIF2AK3 Q9NZJ5 1/20 0.44
HCRTR1 O43613 1/20 0.43
HCRTR2 O43614 1/20 0.43
KAT7 O95251 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
KCNH2 Q12809 1/20 0.41
KAT6B Q8WYB5 1/20 0.41
KAT5 Q92993 1/20 0.41
KAT8 Q9H7Z6 1/20 0.41
LMNA P02545 2/20 0.41
GAA P10253 2/20 0.41
ALDH1A1 P00352 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
ATM Q13315 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5723632 0.92 ECE1 (0.71) ECE1MMEACEKAT6AEIF2AK3
SCHEMBL5723510 0.91 MME (0.59) ECE1MMEACEKAT6ACYP3A4
SCHEMBL5722920 0.90 ECE1 (0.58) ECE1MMEACEKAT6AEIF2AK3
SCHEMBL5722992 0.89 MME (0.57) ECE1MMEACEKAT6AEIF2AK3
SCHEMBL5722993 0.89 MME (0.57) ECE1MMEACEKAT6AEIF2AK3
SCHEMBL5723778 0.86 MME (0.56) ECE1MMEACEKAT6AKAT7
SCHEMBL5723097 0.86 ECE1 (0.67) ECE1MMEACEEIF2AK3HCRTR1
SCHEMBL5723488 0.85 ECE1 (0.66) ECE1MMEACEEIF2AK3HCRTR1
SCHEMBL5723356 0.85 ALDH1A1 (0.51) ECE1MMEACEHCRTR1HCRTR2
SCHEMBL5723398 0.85 ECE1 (0.56) ECE1MMEACEKAT6AEIF2AK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1317428-B1 PYRROLIDINE-2-CARBOXYLIC ACID HYDRAZIDE DERIVATIVES FOR USE AS METALLOPROTEASE INHIBITORS HOFFMANN LA ROCHE (CH) 2006-04-19 EP disclosed