SCHEMBL5724840

SCHEMBL5724840

CCNC1CCCc2onc(O)c21

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
NPC1 O15118 4/20 0.31
RAB9A P51151 4/20 0.31
SMN1; SMN2 Q16637 4/20 0.31
MAPT P10636 2/20 0.31
TP53 P04637 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
HSD17B10 Q99714 1/20 0.30
ESR1 P03372 1/20 0.30
POLB P06746 1/20 0.30
NR4A1 P22736 1/20 0.30
RECQL P46063 1/20 0.30
ESR2 Q92731 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5724843 1.00 CYP1A2 (0.32) CYP1A2CYP2C9NPC1RAB9ASMN1; SMN2
SCHEMBL7983339 0.85 NPC1 (0.34) NPC1RAB9ASMN1; SMN2MAPTTP53
SCHEMBL7983341 0.85 NPC1 (0.34) NPC1RAB9ASMN1; SMN2MAPTTP53
SCHEMBL5725727 0.83 NPC1 (0.33) NPC1RAB9ASMN1; SMN2MAPTTP53
SCHEMBL5724890 0.81 HTR1A (0.32)
SCHEMBL7980246 0.81 HTR1A (0.32)
SCHEMBL7980139 0.78 NPC1 (0.33) NPC1RAB9ASMN1; SMN2MAPTTP53
SCHEMBL7980140 0.78 NPC1 (0.33) NPC1RAB9ASMN1; SMN2MAPTTP53
Bromide SCHEMBL5725876 0.75 LMNA (0.36) CYP2C9NPC1RAB9ASMN1; SMN2KMT2A
Bromide SCHEMBL5725879 0.75 LMNA (0.36) CYP2C9NPC1RAB9ASMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0812318-B1 4-AMINOTETRAHYDROBENZISOXAZOLE OR -ISOTHIAZOLE COMPOUNDS LUNDBECK & CO AS H (DK) 2006-02-08 EP disclosed
US-6174909-B1 FOR TREATING ANALGESIA, PSYCHOSIS, CONVULSIONS, EPILEPSY, ANXIETY, MUSCULAR AND MOVEMENT DISORDERS, SPASTIC DISORDERS OR SYMPTOMS OF HUNTINGTON'S OR PARKINSONS DISEASE H. LUNDBECK A/S (DK) 2001-01-16 US disclosed
US-5998613-A PSYCHOLOGICAL DISORDERS; ANALGESICS; ANTICONVULSANTS H. LUNDBECK A/S (DK) 1999-12-07 US disclosed