SCHEMBL5724985

SCHEMBL5724985

CC(C)(C)OC(=O)NC1CCCc2onc(O)c21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.41
SMN1; SMN2 Q16637 3/20 0.37
LMNA P02545 1/20 0.37
BTK Q06187 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
NFKB1 P19838 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
TP53 P04637 1/20 0.34
MAPT P10636 1/20 0.34
EPHX2 P34913 1/20 0.33
EPHX1 P07099 1/20 0.33
KMT2A Q03164 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CTSK P43235 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5726425 1.00 GAA (0.41) GAASMN1; SMN2LMNABTKHDAC4
SCHEMBL8348647 0.82 GAA (0.38) GAASMN1; SMN2LMNABTKHDAC4
SCHEMBL5724682 0.78 GAA (0.34) GAASMN1; SMN2LMNABTKHDAC4
SCHEMBL5725149 0.74 KDM4D (0.32) SMN1; SMN2LMNA
SCHEMBL5724965 0.74 CHRM3 (0.36) SMN1; SMN2LMNANPC1RAB9ATP53
SCHEMBL24818982 0.72 GAA (0.51) GAABTKNFKB1NFKB2RELA
SCHEMBL764580 0.72 GAA (0.51) GAABTKNFKB1NFKB2RELA
SCHEMBL15192054 0.72 GAA (0.51) GAABTKNFKB1NFKB2RELA
SCHEMBL19667552 0.70 TAS1R3 (0.44) GAALMNAEPHX2KMT2AL3MBTL1
SCHEMBL18735436 0.69 GAA (0.44) GAABTKNFKB1NFKB2RELA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0812318-B1 4-AMINOTETRAHYDROBENZISOXAZOLE OR -ISOTHIAZOLE COMPOUNDS LUNDBECK & CO AS H (DK) 2006-02-08 EP disclosed
US-6174909-B1 FOR TREATING ANALGESIA, PSYCHOSIS, CONVULSIONS, EPILEPSY, ANXIETY, MUSCULAR AND MOVEMENT DISORDERS, SPASTIC DISORDERS OR SYMPTOMS OF HUNTINGTON'S OR PARKINSONS DISEASE H. LUNDBECK A/S (DK) 2001-01-16 US disclosed
US-5998613-A PSYCHOLOGICAL DISORDERS; ANALGESICS; ANTICONVULSANTS H. LUNDBECK A/S (DK) 1999-12-07 US disclosed