SCHEMBL5726753

SCHEMBL5726753

Nc1ccc(C2CCN2C(c2ccccc2)c2ccccc2)c(F)c1O

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 17/20 0.44
OPRK1 P41145 17/20 0.44
OPRL1 P41146 17/20 0.44
OPRD1 P41143 16/20 0.44
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5725406 0.80 OPRM1 (0.38) OPRM1OPRK1OPRL1OPRD1
SCHEMBL5724709 0.73 NPC1 (0.40) ALDH1A1
SCHEMBL5368864 0.64 OPRM1 (0.47) OPRM1OPRK1OPRL1OPRD1ALDH1A1
SCHEMBL11727598 0.63 OPRL1 (0.62) OPRM1OPRK1OPRL1OPRD1
Methane SCHEMBL11728059 0.63 OPRM1 (0.50) OPRM1OPRK1OPRL1OPRD1ALDH1A1
SCHEMBL9792723 0.61 OPRM1 (0.51) OPRM1OPRK1OPRL1OPRD1
SCHEMBL21787342 0.61 OPRM1 (0.51) OPRM1OPRK1OPRL1OPRD1
SCHEMBL13163119 0.61 OPRM1 (0.51) OPRM1OPRK1OPRL1OPRD1
SCHEMBL8534618 0.60 OPRM1 (0.46) OPRM1OPRK1OPRL1OPRD1ALDH1A1
SCHEMBL11461609 0.60 OPRM1 (0.55) OPRM1OPRK1OPRL1OPRD1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1246810-B1 PIPERIDINYLOXY AND PYRROLIDINYLOXYPHENYL OXAZOLIDINONES AS ANTIBACTERIALS ORTHO MCNEIL PHARM INC (US) 2006-05-17 EP disclosed
US-6518285-B2 4-oxo-5-oxazolidineylmethyl derivatives; antibacterials which are active against numerous multidrug-resistant gram positive organisms ORTHO MCNEIL PHARMACEUTICAL, INC. 2003-02-11 US disclosed
US-20020103377-A1 Piperidinyloxy and pyrrolidinyloxy oxazolidinone antibacterials ORTHO-MCNEIL PHARMACEUTICAL, INC. 2002-08-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020103377-A1 Piperidinyloxy and pyrrolidinyloxy oxazolidinone antibacterials OXA1L, RPS27L, RPS27 OPRM1 546/4885OPRK1 1070/4885OPRL1 1129/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.