SCHEMBL5727679

SCHEMBL5727679

CC(C)(C)OC(=O)C1(N)NC(c2ccccc2)C(c2ccccc2)N1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RECQL P46063 1/20 0.40
ABCB1 P08183 1/20 0.39
CHRNA7 P36544 1/20 0.38
NR3C2 P08235 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
LMNA P02545 2/20 0.36
GAA P10253 2/20 0.36
CYP2D6 P10635 1/20 0.35
KDM1A O60341 1/20 0.35
MAOB P27338 1/20 0.35
RORC P51449 2/20 0.34
ALDH1A1 P00352 1/20 0.34
KDM4E B2RXH2 1/20 0.34
TSHR P16473 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
CACNA1F O60840 1/20 0.33
CACNA1D Q01668 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5739111 0.74 AKT1 (0.41) RECQLABCB1
SCHEMBL4924092 0.73 ABCB1 (0.44) RECQLABCB1CHRNA7KDM1AMAOB
SCHEMBL14026296 0.73 ABCB1 (0.44) RECQLABCB1CHRNA7KDM1AMAOB
SCHEMBL13376471 0.73 ABCB1 (0.44) RECQLABCB1CHRNA7KDM1AMAOB
SCHEMBL2764590 0.73 ABCB1 (0.44) RECQLABCB1CHRNA7KDM1AMAOB
SCHEMBL5728175 0.71 GAA (0.44) RECQLGAACYP2D6ALDH1A1KDM4E
SCHEMBL10326487 0.70 RECQL (0.46) RECQLABCB1CHRNA7LMNAGAA
SCHEMBL5728418 0.69 TACR1 (0.36) RECQLABCB1NR3C2LMNAGAA
SCHEMBL7690874 0.69 RAB9A (0.38) ALDH1A1TSHRCACNA1D
SCHEMBL14967416 0.68 L3MBTL1 (0.42) RECQLABCB1KDM1AMAOBRORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1651613-A1 4,5-DIHYDRO-IMIDAZOLE AS P2X7 ION CHANNEL BLOCKERS Aventis Pharmaceuticals, Inc. (US) 2006-05-03 EP disclosed
WO-2005014555-A1 4,5-DIHYDRO-IMIDAZOLE AS P2X7 ION CHANNEL BLOCKERS AVENTIS PHARMACEUTICALS INC. (US) 2005-02-17 WO disclosed