SCHEMBL5727486

SCHEMBL5727486

CC(F)(Cc1cc(F)cc(C#N)c1)CC1CN(C(c2ccccc2)c2ccccc2)C1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 3/20 0.37
SCN9A Q15858 5/20 0.36
SCN5A Q14524 3/20 0.36
OPRD1 P41143 2/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
GLA P06280 1/20 0.35
TSHR P16473 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
P2RX7 Q99572 1/20 0.33
CHRM2 P08172 2/20 0.33
OPRM1 P35372 1/20 0.33
OPRK1 P41145 1/20 0.33
OPRL1 P41146 1/20 0.33
SCN7A Q01118 1/20 0.33
CHRM4 P08173 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4072255 0.91 MEN1 (0.37) MGLLSCN9ASCN5AOPRD1MEN1
SCHEMBL5727242 0.89 OPRM1 (0.36) SCN9ASCN5AOPRD1MEN1KMT2A
SCHEMBL5727699 0.88 CNR1 (0.38) MGLLMEN1KMT2AGLATSHR
SCHEMBL5727552 0.88 SLC6A9 (0.34) MGLLOPRD1MEN1KMT2AGLA
SCHEMBL5727680 0.86 MGLL (0.41) MGLLMEN1KMT2AGLATSHR
SCHEMBL5727357 0.85 P2RX7 (0.35) SCN9ASCN5AOPRD1MEN1KMT2A
SCHEMBL5727485 0.85 TSHR (0.37) MGLLOPRD1MEN1KMT2AGLA
SCHEMBL4686679 0.84 SLC6A9 (0.34) SCN9ASCN5AOPRD1MEN1KMT2A
SCHEMBL5727387 0.84 SLC6A9 (0.34) SCN9ASCN5AOPRD1MEN1KMT2A
SCHEMBL4080122 0.84 CNR1 (0.40) MGLLMEN1KMT2AGLATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1636181-A1 SUBSTITUTED 3-ALKYL AND 3-ALKENYL AZETIDINE DERIVATIVES Merck & Co., Inc. (US) 2006-03-22 EP claimed
WO-2005000809-A1 SUBSTITUTED 3-ALKYL AND 3-ALKENYL AZETIDINE DERIVATIVES MERCK & CO., INC. (US) 2005-01-06 WO claimed