SCHEMBL4072255

SCHEMBL4072255

CC(F)(Cc1cc(F)cc(C#N)c1)CC1CN(C(c2ccc(C#N)cc2)c2cccc(C#N)c2)C1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
TSHR P16473 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
GLA P06280 1/20 0.37
MGLL Q99685 2/20 0.36
ALDH1A1 P00352 3/20 0.35
OPRD1 P41143 1/20 0.34
POLB P06746 1/20 0.34
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NR3C1 P04150 1/20 0.32
NR3C2 P08235 1/20 0.32
TACR1 P25103 1/20 0.31
MRGPRX1 Q96LB2 1/20 0.31
KDM4D Q6B0I6 1/20 0.31
SCN9A Q15858 2/20 0.31
GAA P10253 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5727699 0.94 CNR1 (0.38) MEN1KMT2ATSHRNPSR1GLA
SCHEMBL5727680 0.93 MGLL (0.41) MEN1KMT2ATSHRNPSR1GLA
SCHEMBL4684882 0.92 MEN1 (0.36) MEN1KMT2ATSHRNPSR1GLA
SCHEMBL5727552 0.92 SLC6A9 (0.34) MEN1KMT2ATSHRNPSR1GLA
SCHEMBL5727485 0.91 TSHR (0.37) MEN1KMT2ATSHRNPSR1GLA
SCHEMBL5727486 0.91 MGLL (0.37) MEN1KMT2ATSHRNPSR1GLA
SCHEMBL4080122 0.90 CNR1 (0.40) MEN1KMT2ATSHRNPSR1GLA
SCHEMBL5727631 0.90 MEN1 (0.37) MEN1KMT2ATSHRNPSR1GLA
SCHEMBL4787427 0.86 CNR1 (0.36) MEN1KMT2ATSHRNPSR1GLA
SCHEMBL4681581 0.86 ELANE (0.38) MEN1KMT2ATSHRNPSR1GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2083623-A1 SUBSTITUTED IMIDAZOLES AS BOMBESIN RECEPTOR SUBTYPE-3 MODULATORS Merck & Co., Inc. (US) 2009-08-05 EP disclosed
WO-2008051405-A1 SUBSTITUTED IMIDAZOLES AS BOMBESIN RECEPTOR SUBTYPE-3 MODULATORS MERCK & CO., INC. (US) 2008-05-02 WO disclosed