SCHEMBL5727993

SCHEMBL5727993

COC(=O)Oc1cc(-c2ccc(F)cc2F)sc1NC1CCOCC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 5/20 0.39
GABRA5 P31644 1/20 0.38
JAK2 O60674 1/20 0.38
MAPK14 Q16539 8/20 0.36
GAK O14976 2/20 0.36
RPS6KA4 O75676 1/20 0.36
PRKD3 O94806 1/20 0.36
MAP4K4 O95819 1/20 0.36
MAPK1 P28482 1/20 0.36
MAPK8 P45983 1/20 0.36
MAPK9 P45984 1/20 0.36
CSNK1D P48730 1/20 0.36
RPS6KA3 P51812 1/20 0.36
MAPK10 P53779 1/20 0.36
DDR1 Q08345 1/20 0.36
MAPK11 Q15759 1/20 0.36
TAOK1 Q7L7X3 1/20 0.36
COQ8A Q8NI60 1/20 0.36
PRKD2 Q9BZL6 1/20 0.36
STK36 Q9NRP7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5728276 0.87 CHEK1 (0.40) CHEK1GABRA5JAK2MAPK14GAK
SCHEMBL5728057 0.85 GABRA5 (0.38) CHEK1GABRA5GAKMAPK1
SCHEMBL5434890 0.84 CHEK1 (0.44) CHEK1GABRA5JAK2MAPK14GAK
SCHEMBL5728400 0.75 ACKR3 (0.32) JAK2ACKR3ADORA2A
SCHEMBL5727996 0.75 JAK2 (0.40) CHEK1JAK2
SCHEMBL5728398 0.74 JAK2 (0.38) CHEK1JAK2ADORA2A
SCHEMBL6112105 0.71 ALDH1A1 (0.37) GAKMAPK1MAPK10
SCHEMBL5435719 0.70 IKBKB (0.46) CHEK1JAK2
SCHEMBL5728483 0.69 ACKR3 (0.33) CHEK1JAK2MAPK1ACKR3
SCHEMBL5728485 0.68 ALDH1A1 (0.41) CHEK1MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1694665-A2 SUBSTITUTED THIOPHENES AiCuris GmbH & Co. KG (DE) 2006-08-30 EP disclosed
WO-2005063734-A2 SUBSTITUTED THIOPHENES AICURIS GMBH & CO. KG (DE) 2005-07-14 WO disclosed