SCHEMBL5728485

SCHEMBL5728485

COC(=O)Oc1cc(-c2ccccc2)sc1NC1CCSCC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.41
HPGD P15428 7/20 0.41
KDM4E B2RXH2 5/20 0.41
MAPT P10636 4/20 0.41
GAA P10253 3/20 0.41
HTT P42858 2/20 0.41
TDP1 Q9NUW8 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
ATM Q13315 1/20 0.40
ALOX15 P16050 1/20 0.39
CASP1 P29466 1/20 0.39
CASP7 P55210 1/20 0.39
HSD17B10 Q99714 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
CNR2 P34972 1/20 0.39
CHEK1 O14757 2/20 0.39
TP53 P04637 1/20 0.39
THRB P10828 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2876972 0.82 KDM4E (0.45) ALDH1A1HPGDKDM4EMAPTGAA
SCHEMBL5430057 0.81 CNR2 (0.55) ALDH1A1HPGDKDM4EMAPTGAA
SCHEMBL5730991 0.81 HPGD (0.47) ALDH1A1HPGDKDM4EMAPTGAA
SCHEMBL5728734 0.81 ALDH1A1 (0.47) ALDH1A1HPGDKDM4EMAPTGAA
SCHEMBL5728593 0.80 CHEK1 (0.47) ALDH1A1HPGDKDM4EMAPTGAA
SCHEMBL5728276 0.77 CHEK1 (0.40) KDM4EMAPTTDP1CNR2CHEK1
SCHEMBL2870746 0.74 KDM4E (0.64) ALDH1A1HPGDKDM4EMAPTGAA
SCHEMBL5728057 0.73 GABRA5 (0.38) CHEK1
SCHEMBL5728563 0.72 MAPT (0.61) ALDH1A1HPGDKDM4EMAPTGAA
SCHEMBL5728140 0.71 HPGD (0.42) ALDH1A1HPGDKDM4EMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1694665-A2 SUBSTITUTED THIOPHENES AiCuris GmbH & Co. KG (DE) 2006-08-30 EP disclosed
WO-2005063734-A2 SUBSTITUTED THIOPHENES AICURIS GMBH & CO. KG (DE) 2005-07-14 WO disclosed