SCHEMBL5729079

SCHEMBL5729079

O=C(OCc1ccccc1)N1CCN(NC2CCN(c3ccncc3)CC2)C(=O)C1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 6/20 0.50
CYP2D6 P10635 4/20 0.50
CYP2C9 P11712 4/20 0.50
F10 P00742 1/20 0.45
CYP3A4 P08684 3/20 0.45
SMN1; SMN2 Q16637 2/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
CYP2C19 P33261 1/20 0.43
TMEM97 Q5BJF2 7/20 0.42
SIGMAR1 Q99720 7/20 0.42
HTR1A P08908 2/20 0.42
HRH2 P25021 2/20 0.42
HRH1 P35367 2/20 0.42
HRH3 Q9Y5N1 2/20 0.42
CHRM4 P08173 1/20 0.42
CHRM5 P08912 1/20 0.42
ADRA2A P08913 1/20 0.42
ADRA2B P18089 1/20 0.42
ADRA1D P25100 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5729171 0.81 SMN1; SMN2 (0.51) GRIN2BCYP2D6CYP2C9SMN1; SMN2NPC1
SCHEMBL5729241 0.80 GRIN2B (0.46) GRIN2BCYP2D6CYP2C9F10CYP3A4
SCHEMBL6190799 0.77 ALDH1A1 (0.58) GRIN2BCYP2D6CYP2C9F10SIGMAR1
SCHEMBL1313183 0.75 NPSR1 (0.57) GRIN2BCYP2D6CYP2C9CYP3A4SMN1; SMN2
Hydrochloric Acid SCHEMBL1314129 0.74 MEN1 (0.56) GRIN2BCYP2D6CYP2C9CYP3A4SMN1; SMN2
SCHEMBL29010221 0.74 CYP46A1 (0.54) GRIN2BCYP2D6CYP2C9CYP3A4SMN1; SMN2
SCHEMBL7014966 0.74 ITGB3 (0.52) GRIN2BCYP2D6CYP2C9F10SMN1; SMN2
SCHEMBL6078789 0.72 ITGB3 (0.45) GRIN2BCYP2D6CYP2C9CYP3A4SMN1; SMN2
SCHEMBL9727540 0.71 NPSR1 (0.68) SMN1; SMN2NPC1RAB9ACYP2C19TMEM97
SCHEMBL31461542 0.71 SMN1; SMN2 (0.56) GRIN2BCYP2D6CYP2C9SMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1188755-B1 ACYLHYDRAZINE DERIVATIVES, PROCESS FOR PREPARING THE SAME AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2006-05-03 EP disclosed
US-6723722-B1 BLOOD COAGULATION FACTOR X INHIBITORS; ANTICOAGULANTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2004-04-20 US disclosed
EP-1188755-A1 ACYLHYDRAZINE DERIVATIVES, PROCESS FOR PREPARING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-03-20 EP disclosed