SCHEMBL5729241

SCHEMBL5729241

CN(C1CCN(c2ccncc2)CC1)N1CCN(C(=O)OCc2ccccc2)CC1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 3/20 0.46
CYP2D6 P10635 2/20 0.46
CYP2C9 P11712 2/20 0.46
TMEM97 Q5BJF2 12/20 0.43
SIGMAR1 Q99720 12/20 0.43
HTR1A P08908 3/20 0.42
HRH2 P25021 3/20 0.42
HRH1 P35367 3/20 0.42
HRH3 Q9Y5N1 3/20 0.42
ADRA2A P08913 2/20 0.42
ADRA2B P18089 2/20 0.42
HTR2A P28223 2/20 0.42
HTR2C P28335 2/20 0.42
HTR2B P41595 2/20 0.42
ADRA2C P18825 2/20 0.42
DRD1 P21728 1/20 0.42
HTR1B P28222 1/20 0.42
HTR1E P28566 1/20 0.42
SLC6A4 P31645 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5729666 0.81 SMN1; SMN2 (0.48) SMN1; SMN2NPC1RAB9ACYP2C19MEN1
SCHEMBL5729079 0.80 GRIN2B (0.50) GRIN2BCYP2D6CYP2C9TMEM97SIGMAR1
SCHEMBL20812231 0.78 MEN1 (0.51) TMEM97SIGMAR1HTR1AHRH2HRH1
SCHEMBL803869 0.74 SIGMAR1 (0.51) TMEM97SIGMAR1HTR1AHRH1HRH3
SCHEMBL1313183 0.73 NPSR1 (0.57) GRIN2BCYP2D6CYP2C9TMEM97SIGMAR1
Hydrochloric Acid SCHEMBL1314129 0.72 MEN1 (0.56) GRIN2BCYP2D6CYP2C9TMEM97SIGMAR1
SCHEMBL29010221 0.72 CYP46A1 (0.54) GRIN2BCYP2D6CYP2C9HRH3SMN1; SMN2
SCHEMBL6079558 0.70 ITGB3 (0.44) GRIN2BCYP2D6CYP2C9TMEM97SIGMAR1
SCHEMBL28432287 0.70 MEN1 (0.47) TMEM97SIGMAR1HTR1AHRH2HRH1
SCHEMBL23706353 0.70 SMN1; SMN2 (0.68) GRIN2BCYP2D6CYP2C9TMEM97SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1188755-B1 ACYLHYDRAZINE DERIVATIVES, PROCESS FOR PREPARING THE SAME AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2006-05-03 EP disclosed
US-6723722-B1 BLOOD COAGULATION FACTOR X INHIBITORS; ANTICOAGULANTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2004-04-20 US disclosed
EP-1188755-A1 ACYLHYDRAZINE DERIVATIVES, PROCESS FOR PREPARING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-03-20 EP disclosed