SCHEMBL5729170

SCHEMBL5729170

CC(C)(C)OC(=O)NCCc1cccc(F)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 1/20 0.54
CTSK P43235 1/20 0.54
TAAR1 Q96RJ0 2/20 0.53
CNR1 P21554 1/20 0.51
NQO2 P16083 1/20 0.51
POLB P06746 1/20 0.47
NAMPT P43490 1/20 0.47
IDO1 P14902 1/20 0.47
KDM4E B2RXH2 1/20 0.47
TP53 P04637 1/20 0.46
CA2 P00918 2/20 0.46
OPRM1 P35372 1/20 0.46
OPRD1 P41143 1/20 0.46
OPRK1 P41145 1/20 0.46
CA1 P00915 1/20 0.46
LMNA P02545 1/20 0.45
TSHR P16473 1/20 0.45
PPARG P37231 1/20 0.45
NCOA2 Q15596 1/20 0.45
NCOA1 Q15788 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8401477 0.92 CTSS (0.50) CTSSCTSKTAAR1CNR1NQO2
SCHEMBL5037823 0.90 CTSS (0.48) CTSSCTSKTAAR1CNR1NQO2
SCHEMBL67796 0.89 MAOB (0.54) CTSSCTSKNQO2
SCHEMBL18070221 0.86 CTSK (0.47) CTSSCTSKNQO2POLBNAMPT
SCHEMBL6285264 0.86 CTSS (0.56) CTSSCTSKPOLBLMNATSHR
SCHEMBL31456961 0.86 CTSS (0.56) CTSSCTSKPOLBLMNATSHR
SCHEMBL5117803 0.85 CA1 (0.46) CTSSCTSKNQO2POLBNAMPT
SCHEMBL28321492 0.85 TAAR1 (0.58) TAAR1CNR1POLBTP53OPRM1
SCHEMBL8399573 0.85 GPR119 (0.53) CTSSCTSKNQO2NAMPTIDO1
SCHEMBL18198086 0.85 CTSS (0.54) CTSSCTSKNQO2IDO1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720836-A1 6-SUBSTITUTED 2,3,4,5-TETRAHYDRO-1H-BENZO [D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS ELI LILLY AND COMPANY (US) 2006-11-15 EP disclosed
WO-2005082859-A1 6-SUBSTITUTED 2,3,4,5-TETRAHYDRO-1H-BENZO[D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS ELI LILLY AND COMPANY (US) 2005-09-09 WO disclosed