SCHEMBL5729581

SCHEMBL5729581

C=CC(C)(C)CCc1ccc(C#N)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.46
LOXL2 Q9Y4K0 2/20 0.43
TSHR P16473 1/20 0.42
HSD17B10 Q99714 1/20 0.42
KCNJ1 P48048 1/20 0.42
KCNH2 Q12809 1/20 0.42
KIF11 P52732 1/20 0.38
HRH3 Q9Y5N1 1/20 0.37
MAOA P21397 2/20 0.37
MAOB P27338 2/20 0.37
ALDH1A1 P00352 1/20 0.36
EPHX2 P34913 1/20 0.36
DAO P14920 2/20 0.36
NPC1 O15118 1/20 0.36
GAA P10253 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
PPARD Q03181 2/20 0.35
PPARA Q07869 2/20 0.35
CYP19A1 P11511 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11910300 0.80 CYP2A6 (0.54) CYP2A6LOXL2TSHRHSD17B10KCNJ1
SCHEMBL7922825 0.77 LOXL2 (0.50) CYP2A6LOXL2TSHRHSD17B10KCNJ1
SCHEMBL8995507 0.77 CYP2A6 (0.50) CYP2A6LOXL2TSHRHSD17B10KCNJ1
SCHEMBL5410448 0.77 GFER (0.48) CYP2A6LOXL2TSHRMAOAMAOB
SCHEMBL5419014 0.76 AOC3 (0.41) CYP2A6LOXL2HSD17B10ALDH1A1SMN1; SMN2
SCHEMBL29065555 0.73 TSHR (0.54) CYP2A6LOXL2TSHRHSD17B10KCNJ1
SCHEMBL1004267 0.72 LOXL2 (0.64) CYP2A6LOXL2TSHRHSD17B10KCNJ1
SCHEMBL2968409 0.72 KCNJ1 (0.48) CYP2A6LOXL2TSHRHSD17B10KCNJ1
SCHEMBL18560067 0.72 KCNJ1 (0.48) CYP2A6LOXL2TSHRHSD17B10KCNJ1
SCHEMBL14460154 0.71 TSHR (0.57) CYP2A6LOXL2TSHRHSD17B10KCNJ1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720836-A1 6-SUBSTITUTED 2,3,4,5-TETRAHYDRO-1H-BENZO [D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS ELI LILLY AND COMPANY (US) 2006-11-15 EP disclosed
WO-2005082859-A1 6-SUBSTITUTED 2,3,4,5-TETRAHYDRO-1H-BENZO[D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS ELI LILLY AND COMPANY (US) 2005-09-09 WO disclosed