SCHEMBL5730809

SCHEMBL5730809

O=C(NCc1[c]c(OCCCCOc2cccc(-c3ccccc3)c2)ccc1)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 4/20 0.47
HDAC1 Q13547 2/20 0.46
HDAC2 Q92769 2/20 0.46
MRGPRX4 Q96LA9 1/20 0.46
NPC1 O15118 1/20 0.45
HPGD P15428 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
HRH3 Q9Y5N1 6/20 0.45
F10 P00742 1/20 0.45
MAOB P27338 1/20 0.44
EPHX2 P34913 1/20 0.43
NR4A2 P43354 1/20 0.43
PPARG P37231 1/20 0.42
PPARD Q03181 1/20 0.42
PPARA Q07869 1/20 0.42
ROCK2 O75116 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5730910 0.98 NR1H4 (0.45) NR1H4HDAC1HDAC2MRGPRX4NPC1
SCHEMBL5730552 0.91 NPC1 (0.47) NR1H4HDAC1HDAC2NPC1HPGD
SCHEMBL5353021 0.89 NPC1 (0.47) NR1H4HDAC1HDAC2NPC1HPGD
SCHEMBL5730023 0.87 HPGD (0.50) NR1H4NPC1HPGDRAB9ASMN1; SMN2
SCHEMBL5731178 0.83 HPGD (0.51) NR1H4NPC1HPGDRAB9ASMN1; SMN2
SCHEMBL5729685 0.81 NQO2 (0.47) NPC1HPGDRAB9ASMN1; SMN2EPHX2
SCHEMBL4894779 0.74 FFAR4 (0.50) NR1H4HDAC1HDAC2EPHX2PPARG
SCHEMBL4885499 0.72 FFAR4 (0.50) NR1H4HDAC1HDAC2PPARGPPARD
SCHEMBL7044733 0.69 FFAR4 (0.72) HDAC1HDAC2MRGPRX4HRH3PPARA
SCHEMBL5729898 0.69 PPARA (0.42) NPC1HPGDRAB9APPARGPPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1401434-B1 MODULATORS OF PEROXISOME PROLIFERATOR ACTIVATED RECEPTORS (PPAR) LILLY CO ELI (US) 2006-11-15 EP disclosed