SCHEMBL5732043

SCHEMBL5732043

Brc1ccccc1CSC1=NCCN1

nearest known ligand 0.67

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.67
LMNA P02545 1/20 0.67
GFER P55789 3/20 0.51
CYP2D6 P10635 3/20 0.48
MAPT P10636 3/20 0.48
CYP3A4 P08684 2/20 0.48
CYP1A2 P05177 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
RAB9A P51151 1/20 0.48
HIF1A Q16665 1/20 0.48
NISCH Q9Y2I1 1/20 0.43
HTR1A P08908 1/20 0.42
ADRA2A P08913 1/20 0.42
ADRA2B P18089 1/20 0.42
ADRA2C P18825 1/20 0.42
ALDH1A1 P00352 1/20 0.41
CDC7 O00311 1/20 0.41
DBF4 Q9UBU7 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5731969 0.81 KMT2A (0.67) KMT2ALMNAGFERCYP2D6MAPT
SCHEMBL5733176 0.81 KMT2A (0.97) KMT2ALMNAGFERCYP2D6MAPT
SCHEMBL5731047 0.81 KMT2A (0.67) KMT2ALMNAGFERCYP2D6MAPT
SCHEMBL2493368 0.81 KMT2A (0.67) KMT2ALMNAGFERCYP2D6MAPT
Bromide SCHEMBL3176423 0.80 KMT2A (0.65) KMT2ALMNAGFERCYP2D6MAPT
Hydrochloric Acid SCHEMBL2493369 0.80 KMT2A (0.69) KMT2ALMNAGFERCYP2D6MAPT
SCHEMBL3163430 0.77 MAPT (0.65) KMT2ALMNAGFERCYP2D6MAPT
Hydrochloric Acid SCHEMBL3180041 0.76 KMT2A (0.63) KMT2ALMNAGFERCYP2D6MAPT
SCHEMBL5731245 0.75 KMT2A (0.58) KMT2ALMNAGFERCYP2D6MAPT
SCHEMBL5732498 0.74 MAPT (0.66) KMT2ALMNAGFERCYP2D6MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1651613-A1 4,5-DIHYDRO-IMIDAZOLE AS P2X7 ION CHANNEL BLOCKERS Aventis Pharmaceuticals, Inc. (US) 2006-05-03 EP disclosed
WO-2005014555-A1 4,5-DIHYDRO-IMIDAZOLE AS P2X7 ION CHANNEL BLOCKERS AVENTIS PHARMACEUTICALS INC. (US) 2005-02-17 WO disclosed