SCHEMBL5732347

SCHEMBL5732347

CC(CCOc1ccc(CN)cc1)(S(C)(=O)=O)S(C)(=O)=O

nearest known ligand 0.49

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.49
NFE2L2 Q16236 1/20 0.49
MAOB P27338 3/20 0.41
S1PR1 P21453 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL506565 0.80 KEAP1 (0.58) KEAP1NFE2L2MAOB
SCHEMBL7973439 0.73 KEAP1 (0.67) KEAP1NFE2L2MAOB
SCHEMBL7988040 0.71 KEAP1 (0.64) KEAP1NFE2L2MAOB
SCHEMBL7388158 0.71 KEAP1 (0.64) KEAP1NFE2L2MAOB
SCHEMBL2911524 0.70 KEAP1 (0.63) KEAP1NFE2L2MAOB
SCHEMBL1157194 0.70 KEAP1 (0.63) KEAP1NFE2L2MAOB
SCHEMBL23905132 0.69 LTA4H (0.64) KEAP1NFE2L2MAOB
SCHEMBL7983918 0.69 KEAP1 (0.62) KEAP1NFE2L2MAOB
SCHEMBL12990053 0.69 KEAP1 (0.62) KEAP1NFE2L2MAOB
SCHEMBL12408533 0.69 KEAP1 (0.62) KEAP1NFE2L2MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720836-A1 6-SUBSTITUTED 2,3,4,5-TETRAHYDRO-1H-BENZO [D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS ELI LILLY AND COMPANY (US) 2006-11-15 EP disclosed
WO-2005082859-A1 6-SUBSTITUTED 2,3,4,5-TETRAHYDRO-1H-BENZO[D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS ELI LILLY AND COMPANY (US) 2005-09-09 WO disclosed