SCHEMBL5733402

SCHEMBL5733402

NC(=O)c1ccc2[nH]c(N3CCC(Cl)(Cc4ccccc4)CC3)cc2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 5/20 0.44
SLC6A4 P31645 5/20 0.44
SLC6A3 Q01959 5/20 0.44
CYP2D6 P10635 1/20 0.44
F2 P00734 2/20 0.41
CHEK1 O14757 2/20 0.39
MMP2 P08253 1/20 0.38
MMP13 P45452 1/20 0.38
CHEK2 O96017 3/20 0.37
GAA P10253 1/20 0.37
NPY5R Q15761 1/20 0.37
OPRK1 P41145 2/20 0.37
OPRM1 P35372 1/20 0.37
OPRD1 P41143 1/20 0.37
KCNH2 Q12809 1/20 0.37
GRIN2D O15399 1/20 0.37
GRIN3B O60391 1/20 0.37
GRIN1 Q05586 1/20 0.37
GRIN2A Q12879 1/20 0.37
GRIN2B Q13224 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5203581 0.81 GAA (0.54) CHEK1GAAGRIN2DGRIN3BGRIN1
SCHEMBL7375633 0.76 CHEK1 (0.50) CHEK1MMP2MMP13CHEK2GAA
SCHEMBL5733310 0.75 GAA (0.44) SLC6A2SLC6A4CHEK1CHEK2GAA
SCHEMBL5733400 0.74 ROCK2 (0.41) SLC6A2SLC6A4SLC6A3CYP2D6F2
SCHEMBL5734927 0.73 CHEK1 (0.41) F2CHEK1MMP2MMP13CHEK2
SCHEMBL5369135 0.73 CHEK1 (0.52) CHEK1CHEK2OPRK1OPRM1
SCHEMBL5374691 0.73 GAA (0.47) CHEK1CHEK2GAAGRIN2DGRIN3B
SCHEMBL5733660 0.72 GAA (0.54) CHEK2GAAGRIN2DGRIN3BGRIN1
SCHEMBL5732647 0.72 GAA (0.48) SLC6A2SLC6A4SLC6A3CHEK1CHEK2
SCHEMBL5374221 0.70 GAA (0.46) SLC6A2SLC6A4SLC6A3CHEK1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1080078-B1 HETEROCYCLIC COMPOUNDS AND METHODS TO TREAT CARDIAC FAILURE AND OTHER DISORDERS SCIOS INC (US) 2006-02-01 EP claimed