SCHEMBL5734016

SCHEMBL5734016

C=CS(=O)(=O)N1CCNCC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.46
F13A1 P00488 1/20 0.38
TGM2 P21980 1/20 0.38
TGM1 P22735 1/20 0.38
MAPT P10636 1/20 0.37
USP2 O75604 1/20 0.34
ALDH1A1 P00352 2/20 0.33
PKM P14618 1/20 0.33
KMT2A Q03164 2/20 0.32
BTK Q06187 1/20 0.31
LMNA P02545 1/20 0.30
CYP3A4 P08684 1/20 0.30
GABRA1 P14867 1/20 0.30
TSHR P16473 1/20 0.30
GABRG2 P18507 1/20 0.30
NFKB1 P19838 1/20 0.30
GABRB3 P28472 1/20 0.30
GABRA5 P31644 1/20 0.30
GABRA3 P34903 1/20 0.30
GABRA2 P47869 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL23389815 0.98 KDM4E (0.45) KDM4EF13A1TGM2TGM1MAPT
SCHEMBL28831827 0.86 KDM4E (0.39) KDM4EF13A1TGM2TGM1MAPT
SCHEMBL20546681 0.82 POLB (0.35) KMT2ABTKTSHRSMYD3
SCHEMBL10803979 0.82
SCHEMBL13970069 0.82 POLB (0.35) KMT2ABTKTSHRSMYD3
SCHEMBL4256096 0.77 CA1 (0.43) KDM4EF13A1TGM2TGM1USP2
SCHEMBL3598091 0.76 KDM4E (0.46) KDM4EF13A1TGM2TGM1MAPT
SCHEMBL2428756 0.75 CA1 (0.48) KDM4EF13A1TGM2TGM1MAPT
SCHEMBL3548115 0.72 KDM4E (0.52) KDM4EF13A1TGM2TGM1MAPT
SCHEMBL3554550 0.71 SMYD3 (0.33) SMYD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111499313-B Cement-based aerogel heat insulation board and preparation method thereof 贵州航天建设工程有限公司 2024-08-09 CN claimed
CN-111499313-A Cement-based aerogel heat-insulation plate and preparation method thereof 贵州航天建设工程有限公司 2020-08-07 CN claimed
EP-4637926-A1 SYNTHESIS, PHARMACOLOGY AND USE OF NEW WATER-SOLUBLE AND SELECTIVE FMS-LIKE TYROSINE KINASE 3 (FLT3) INHIBITORS Universität Regensburg (DE) 2025-10-29 EP disclosed
CN-111499313-B Cement-based aerogel heat insulation board and preparation method thereof 贵州航天建设工程有限公司 2024-08-09 CN disclosed
WO-2024132278-A1 SYNTHESIS, PHARMACOLOGY AND USE OF NEW WATER-SOLUBLE AND SELECTIVE FMS-LIKE TYROSINE KINASE 3 (FLT3) INHIBITORS UNIVERSITÄT REGENSBURG (DE) 2024-06-27 WO disclosed
WO-2024132278-A1 SYNTHESIS, PHARMACOLOGY AND USE OF NEW WATER-SOLUBLE AND SELECTIVE FMS-LIKE TYROSINE KINASE 3 (FLT3) INHIBITORS UNIVERSITÄT REGENSBURG (DE) 2024-06-27 WO disclosed
EP-4389223-A1 SYNTHESIS, PHARMACOLOGY AND USE OF NEW WATER-SOLUBLE AND SELECTIVE FMS-LIKE TYROSINE KINASE 3 (FLT3) INHIBITORS Universität Regensburg (DE) 2024-06-26 EP disclosed
US-20230052528-A1 TASPASE1 INHIBITORS AND USES THEREOF UNIV CALIFORNIA (US) 2023-02-16 US disclosed
CN-115397818-A Aminopyrimidine derivatives and their use as modulators of arene receptors 东亚ST株式会社 2022-11-25 CN disclosed
WO-2021102359-A2 TASPASE1 INHIBITORS AND USES THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-05-27 WO disclosed
CN-111499313-A Cement-based aerogel heat-insulation plate and preparation method thereof 贵州航天建设工程有限公司 2020-08-07 CN disclosed
EP-2029606-B1 CYCLOPROPYL FUSED INDOLOBENZAZEPINE HCV NS5B INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2010-05-26 EP disclosed
EP-0986551-B1 SULFONAMIDE DERIVATIVES, THEIR PRODUCTION AND USE TAKEDA PHARMACEUTICAL (JP) 2006-08-02 EP disclosed
US-6359134-B1 ANTICOAGULANTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-03-19 US disclosed
EP-0986551-A1 SULFONAMIDE DERIVATIVES, THEIR PRODUCTION AND USE Takeda Pharmaceutical Company Limited (JP) 2000-03-22 EP disclosed
WO-1998054164-A1 SULFONAMIDE DERIVATIVES, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-12-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230052528-A1 TASPASE1 INHIBITORS AND USES THEREOF RNASE1, TASP1, TPP1 KDM4E 3697/4885F13A1 4092/4885TGM2 209/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.