SCHEMBL5735392

SCHEMBL5735392

C[C@H]1OC(=O)N(Cc2ccccc2)[C@@H]1C(=O)OCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
FOLH1 Q04609 2/20 0.41
ELANE P08246 2/20 0.41
GRM2 Q14416 1/20 0.41
NAAA Q02083 1/20 0.41
TSHR P16473 1/20 0.41
CACNA1G O43497 1/20 0.41
CACNA1H O95180 1/20 0.41
CACNA1I Q9P0X4 1/20 0.41
HTR2C P28335 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
FABP7 O15540 1/20 0.40
FABP5 Q01469 1/20 0.40
FKBP1A P62942 1/20 0.40
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5735391 1.00 ALDH1A1 (0.42) ALDH1A1FOLH1ELANEGRM2NAAA
SCHEMBL21584135 0.87 TDP1 (0.50) ALDH1A1TSHRTDP1FKBP1A
SCHEMBL5734544 0.84 ALDH1A1 (0.44) ALDH1A1FOLH1ELANENAAATSHR
SCHEMBL5734541 0.84 ALDH1A1 (0.44) ALDH1A1FOLH1ELANENAAATSHR
SCHEMBL5733366 0.84 EHMT2 (0.42) ALDH1A1GRM2TDP1
SCHEMBL5733370 0.84 EHMT2 (0.42) ALDH1A1GRM2TDP1
SCHEMBL5736768 0.83 FKBP1A (0.38) ALDH1A1FOLH1ELANENAAATSHR
SCHEMBL5736762 0.83 FKBP1A (0.38) ALDH1A1FOLH1ELANENAAATSHR
SCHEMBL5735748 0.83 ELANE (0.38) ALDH1A1FOLH1ELANENAAATSHR
SCHEMBL5735745 0.83 ELANE (0.38) ALDH1A1FOLH1ELANENAAATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0933379-B1 NOVEL PEPTIDE DERIVATIVES HAVING THIAZOLYL-ALANINE RESIDUE SHIONOGI & CO (JP) 2006-03-22 EP disclosed
US-6319902-B1 TO ACTIVATE THE CENTRAL NERVOUS SYSTEM, SUCH AS, FOR EXAMPLE, SUSTAINED ACETYLCHOLINE RELEASING ACTION, ANTI-RESERPINE ACTION AND LOCOMOTOR INCREMENT SHIONOGI & CO., LTD. (JP) 2001-11-20 US disclosed
EP-0933379-A1 NOVEL PEPTIDE DERIVATIVES HAVING THIAZOLYL-ALANINE RESIDUE SHIONOGI & CO., LTD. (JP) 1999-08-04 EP disclosed